SCHEMBL30451127

SCHEMBL30451127

COc1ccc(CN2Cc3cc(F)ccc3C2=O)c(OC)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.48
GRIN2B Q13224 1/20 0.46
KDM4E B2RXH2 2/20 0.45
P2RX7 Q99572 4/20 0.44
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HDAC9 Q9UKV0 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44
EGLN1 Q9GZT9 1/20 0.43
ADAM17 P78536 2/20 0.43
DRD2 P14416 1/20 0.42
DRD4 P21917 1/20 0.42
DRD3 P35462 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2144643 0.86 KDM4E (0.45) GRIN2BKDM4EHDAC3HDAC4HDAC1
SCHEMBL1530558 0.86 HDAC3 (0.46) GRIN2BKDM4EHDAC3HDAC4HDAC1
SCHEMBL14991601 0.83 LMNA (0.49) ADAM17LMNA
SCHEMBL2144806 0.82 KMT2A (0.46) KDM4EHDAC3HDAC4HDAC1HDAC7
SCHEMBL7271173 0.81 TACR1 (0.44) TACR1KDM4EP2RX7HDAC3HDAC4
SCHEMBL1530198 0.79 WIZ (0.41) GRIN2BKDM4EHDAC3HDAC4HDAC1
SCHEMBL30874421 0.79 EGLN1 (0.50) KDM4EHDAC3HDAC4HDAC1HDAC7
SCHEMBL30059679 0.79 HDAC3 (0.44) TACR1KDM4EHDAC3HDAC4HDAC1
SCHEMBL22226371 0.79 EGLN1 (0.50) KDM4EHDAC3HDAC4HDAC1HDAC7
SCHEMBL27721893 0.78 HDAC3 (0.48) TACR1KDM4EHDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116261562-A PI 3K-alpha inhibitors and methods of use thereof 传达治疗有限公司 2023-06-13 CN disclosed