SCHEMBL30451246

SCHEMBL30451246

[2H]c1c(CC(N)=O)cccc1NC(=O)c1cc(F)cc(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.45
P2RX1 P51575 2/20 0.45
RHOC P08134 2/20 0.45
RHOA P61586 2/20 0.45
PTGS1 P23219 3/20 0.45
MAPT P10636 2/20 0.44
MEN1 O00255 2/20 0.44
RAB9A P51151 2/20 0.44
KMT2A Q03164 2/20 0.44
ABL1 P00519 1/20 0.44
BCR P11274 1/20 0.44
NPC1 O15118 1/20 0.44
KCNK3 O14649 1/20 0.44
RPS6KB1 P23443 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
HTT P42858 1/20 0.42
HDAC3 O15379 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
TRPA1 O75762 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23985109 0.90 NR1H4 (0.51) LMNAP2RX1RHOCRHOAPTGS1
SCHEMBL23985155 0.79 KCNK3 (0.58) LMNAP2RX1RHOCRHOAPTGS1
SCHEMBL23985152 0.78 RHOC (0.60) LMNAP2RX1RHOCRHOAPTGS1
SCHEMBL30554615 0.73 P2RX1 (0.65) P2RX1RHOCRHOAMAPTRXFP1
SCHEMBL3246188 0.73 P2RX1 (0.65) P2RX1RHOCRHOAMAPTRXFP1
SCHEMBL678377 0.72 PTGS1 (0.68) LMNAP2RX1RHOCRHOAPTGS1
Hydrochloric Acid SCHEMBL30481169 0.71 EPHX1 (0.44) MAPTMEN1KMT2A
SCHEMBL22772371 0.71 ABL1 (0.57) LMNAP2RX1RHOCRHOAPTGS1
SCHEMBL5389064 0.70 RXRA (0.49)
SCHEMBL14528862 0.69 RHOC (0.48) RHOCRHOAHDAC3HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116261562-A PI 3K-alpha inhibitors and methods of use thereof 传达治疗有限公司 2023-06-13 CN disclosed