SCHEMBL30451293

SCHEMBL30451293

Cc1nnc(N)c2ccc(-c3cc(B(O)O)cc4ccoc34)cc12

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PLG P00747 1/20 0.36
F12 P00748 1/20 0.36
F11 P03951 1/20 0.36
KLKB1 P03952 1/20 0.36
PRSS1 P07477 1/20 0.36
PRSS2 P07478 1/20 0.36
PRSS3 P35030 1/20 0.36
SLC22A12 Q96S37 4/20 0.31
XDH P47989 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24252383 1.00 PLG (0.36) PLGF12F11KLKB1PRSS1
SCHEMBL26771276 0.92 PLG (0.31) PLGF12F11KLKB1PRSS1
SCHEMBL24252263 0.77 MAP4K4 (0.37) PLGF12F11KLKB1PRSS1
SCHEMBL24252648 0.77 PLG (0.31) PLGF12F11KLKB1PRSS1
SCHEMBL24252292 0.76 PLG (0.34) PLGF12F11KLKB1PRSS1
SCHEMBL24252506 0.75 MAP4K4 (0.37) PLGF12F11KLKB1PRSS1
SCHEMBL24252659 0.75 DHFR (0.31) PLGF12F11KLKB1PRSS1
SCHEMBL24252733 0.74 PLG (0.56) PLGF12F11KLKB1PRSS1
SCHEMBL30451657 0.74 PLG (0.56) PLGF12F11KLKB1PRSS1
SCHEMBL24252663 0.74 PLG (0.33) PLGF12F11KLKB1PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116947903-A Inhibitors of complement factors and uses thereof 安尼艾克松股份有限公司 2023-10-27 CN disclosed
CN-116261564-A Inhibitors of complement factors and uses thereof 安尼艾克松股份有限公司 2023-06-13 CN disclosed
EP-4185592-A1 INHIBITORS OF COMPLEMENT FACTORS AND USES THEREOF Annexon, Inc. (US) 2023-05-31 EP disclosed