SCHEMBL30453478

SCHEMBL30453478

NC(=O)c1ccc(N2CCC3(CC2)CC(=O)C3)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 6/20 0.48
ITGA2B P08514 6/20 0.48
CHRNA7 P36544 1/20 0.48
CHRNA10 Q9GZZ6 1/20 0.48
CHRNA9 Q9UGM1 1/20 0.48
F2 P00734 2/20 0.46
PRSS1 P07477 2/20 0.46
PRSS2 P07478 2/20 0.46
PRSS3 P35030 2/20 0.46
TMPRSS6 Q8IU80 2/20 0.46
ST14 Q9Y5Y6 2/20 0.46
GRIN2D O15399 1/20 0.42
GRIN3B O60391 1/20 0.42
GRIN1 Q05586 1/20 0.42
GRIN2A Q12879 1/20 0.42
GRIN2B Q13224 1/20 0.42
GRIN2C Q14957 1/20 0.42
GRIN3A Q8TCU5 1/20 0.42
CYP3A4 P08684 3/20 0.42
CHEK1 O14757 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22904552 0.88 ITGB3 (0.46) ITGB3ITGA2BCHRNA7CHRNA10CHRNA9
SCHEMBL30078285 0.86 KDM4E (0.53) ITGB3ITGA2BCYP3A4CHEK1USP2
SCHEMBL26648503 0.81 ALDH1A1 (0.57) CYP3A4USP2ALDH1A1CYP2C19CYP1A2
SCHEMBL24832881 0.80 ALDH1A1 (0.48) ITGB3ITGA2BCYP3A4USP2ALDH1A1
SCHEMBL377181 0.79 CHRNA7 (0.55) ITGB3ITGA2BCHRNA7CHRNA10CHRNA9
SCHEMBL1377551 0.78 CHRNA7 (0.54) ITGB3ITGA2BCHRNA7CHRNA10CHRNA9
SCHEMBL3883363 0.76 MAPT (0.61) CHRNA7CHRNA10CHRNA9F2PRSS1
SCHEMBL4131556 0.76 HRH3 (0.60) ITGB3ITGA2BCHRNA7CHRNA10CHRNA9
SCHEMBL1397421 0.74 NPC1 (0.61) CHRNA7CHRNA10CHRNA9F2PRSS1
SCHEMBL4873981 0.74 NPC1 (0.61) CHRNA7CHRNA10CHRNA9F2PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023121713-A1 BCL-2 INHIBITORS NEW AVE PHARMACEUTICAL INC. (US) 2023-06-29 WO disclosed
WO-2023122000-A1 BCL-2 INHIBITORS NEWAVE PHARMACEUTICAL INC. (US) 2023-06-29 WO disclosed