SCHEMBL30454449

SCHEMBL30454449

COc1ccc(-c2ccc3nc(C)[nH]c(=O)c3c2)cc1CC(=O)N(C)C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.49
HSD17B10 Q99714 2/20 0.49
LMNA P02545 1/20 0.49
TRPV1 Q8NER1 3/20 0.47
POLB P06746 4/20 0.46
NPSR1 Q6W5P4 1/20 0.46
ACVR1 Q04771 2/20 0.42
ROCK2 O75116 2/20 0.41
GUSB P08236 2/20 0.40
CYP1A1 P04798 1/20 0.40
CYP1B1 Q16678 1/20 0.40
IP6K1 Q92551 1/20 0.39
MMP13 P45452 1/20 0.39
TYMS P04818 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
TSHR P16473 1/20 0.39
ALDH1A1 P00352 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30454826 0.92 HSD17B10 (0.49) KDM4EHSD17B10LMNATRPV1POLB
SCHEMBL30455167 0.86 HSD17B10 (0.48) KDM4EHSD17B10LMNATRPV1POLB
SCHEMBL30455646 0.81 RXFP1 (0.40) KDM4EHSD17B10LMNAPOLBMEN1
SCHEMBL29002507 0.74 HSD17B10 (0.46) KDM4EHSD17B10LMNATRPV1POLB
SCHEMBL30594962 0.72 NPC1 (0.41) KDM4EHSD17B10LMNAPOLBMEN1
SCHEMBL30455110 0.72 AMY1A (0.39) KDM4EHSD17B10LMNAPOLBNPSR1
SCHEMBL30594977 0.72 POLB (0.42) KDM4EHSD17B10LMNAPOLBMEN1
SCHEMBL30455089 0.70 AMY1A (0.39) KDM4EHSD17B10LMNAPOLBNPSR1
SCHEMBL24802434 0.70 MAPK8 (0.48) HSD17B10POLBMEN1KMT2ATSHR
SCHEMBL1257374 0.67 KDM4E (1.00) KDM4EHSD17B10LMNATRPV1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116143708-A Polysubstituted benzazepine heteroaryl derivative and application thereof 四川汇宇制药股份有限公司 2023-05-23 CN disclosed