SCHEMBL30454826

SCHEMBL30454826

COc1cc(-c2ccc3nc(C)[nH]c(=O)c3c2)ccc1CC(=O)N(C)C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.49
KDM4E B2RXH2 2/20 0.49
LMNA P02545 1/20 0.49
TRPV1 Q8NER1 5/20 0.47
POLB P06746 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
AMY1A P0DUB6 1/20 0.44
ACVR1 Q04771 2/20 0.42
ROCK2 O75116 1/20 0.41
CYP1A1 P04798 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP1B1 Q16678 1/20 0.40
GUSB P08236 1/20 0.39
IP6K1 Q92551 1/20 0.39
MMP13 P45452 1/20 0.39
CHEK1 O14757 1/20 0.39
TYMS P04818 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
MEN1 O00255 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30454449 0.92 KDM4E (0.49) HSD17B10KDM4ELMNATRPV1POLB
SCHEMBL30455167 0.84 HSD17B10 (0.48) HSD17B10KDM4ELMNATRPV1POLB
SCHEMBL30594962 0.81 NPC1 (0.41) HSD17B10KDM4ELMNAPOLBAMY1A
SCHEMBL30594977 0.80 POLB (0.42) HSD17B10KDM4ELMNAPOLBAMY1A
SCHEMBL30455110 0.80 AMY1A (0.39) HSD17B10KDM4ELMNAPOLBNPSR1
SCHEMBL30455089 0.79 AMY1A (0.39) HSD17B10KDM4ELMNAPOLBNPSR1
SCHEMBL30455313 0.77 TRPV1 (0.47) HSD17B10KDM4ELMNATRPV1POLB
SCHEMBL29002513 0.77 TRPV1 (0.47) HSD17B10KDM4ELMNATRPV1POLB
SCHEMBL29002507 0.74 HSD17B10 (0.46) HSD17B10KDM4ELMNATRPV1POLB
SCHEMBL30455646 0.72 RXFP1 (0.40) HSD17B10KDM4ELMNAPOLBCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116143708-A Polysubstituted benzazepine heteroaryl derivative and application thereof 四川汇宇制药股份有限公司 2023-05-23 CN disclosed