SCHEMBL30454529

SCHEMBL30454529

COC(=O)c1c[nH]c(/C=C2\C(=O)Nc3ccc(F)cc32)c1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 2/20 0.60
AKT2 P31751 3/20 0.54
CCNE1 P24864 2/20 0.54
CDK2 P24941 2/20 0.54
CCNE2 O96020 1/20 0.54
TLK2 Q86UE8 3/20 0.51
AURKA O14965 1/20 0.51
RAF1 P04049 1/20 0.51
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
FLT3 P36888 2/20 0.48
KDR P35968 1/20 0.48
ALK Q9UM73 1/20 0.48
NTRK1 P04629 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30453243 0.87 PDPK1 (0.60) PDPK1AKT2AURKARAF1MEN1
SCHEMBL3799498 0.86 AKT2 (0.67) PDPK1AKT2CCNE1CDK2CCNE2
SCHEMBL31216363 0.79 KDR (0.71) PDPK1AKT2TLK2AURKAMEN1
SCHEMBL2114561 0.79 PAK4 (0.57) PDPK1AKT2TLK2AURKAMEN1
SCHEMBL1965178 0.78 AURKA (0.69) PDPK1TLK2AURKARAF1MEN1
SCHEMBL12580695 0.78 AURKA (0.69) PDPK1TLK2AURKARAF1MEN1
SCHEMBL2115629 0.78 AKT2 (0.53) PDPK1AKT2TLK2AURKAMEN1
SCHEMBL5728671 0.75 PDPK1 (1.00) PDPK1TLK2KDRNTRK1
SCHEMBL5361523 0.75 PDPK1 (1.00) PDPK1TLK2KDRNTRK1
SCHEMBL3284152 0.74 FLT3 (0.68) PDPK1CCNE1CDK2CCNE2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113181362-B Medicament for preventing and/or treating amyotrophic lateral sclerosis 国立大学法人京都大学 2023-06-13 CN disclosed