SCHEMBL30456978

SCHEMBL30456978

COC(=O)c1cc(C(=O)O)ccc1OC

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.65
CA1 P00915 1/20 0.65
CA2 P00918 1/20 0.65
CA4 P22748 1/20 0.65
CA6 P23280 1/20 0.65
CA7 P43166 1/20 0.65
TPMT P51580 1/20 0.65
CA9 Q16790 1/20 0.65
CA14 Q9ULX7 1/20 0.65
HTT P42858 3/20 0.59
LMNA P02545 3/20 0.59
RAB9A P51151 2/20 0.59
MAPK1 P28482 1/20 0.59
TSHR P16473 2/20 0.56
ALDH1A1 P00352 2/20 0.55
TTR P02766 1/20 0.53
PKM P14618 1/20 0.53
MAPT P10636 2/20 0.51
KDM4E B2RXH2 2/20 0.51
NPSR1 Q6W5P4 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5168276 1.00 CA12 (0.65) CA12CA1CA2CA4CA6
SCHEMBL5169870 0.89 MAPT (0.64) CA12CA1CA2CA7CA9
SCHEMBL29678875 0.89 MAPT (0.64) CA12CA1CA2CA7CA9
SCHEMBL6931187 0.87 CYP1A2 (0.63) HTTLMNATSHRALDH1A1MAPT
SCHEMBL29446743 0.87 CA12 (0.71) CA12CA1CA2CA4CA6
SCHEMBL901309 0.87 CA12 (0.71) CA12CA1CA2CA4CA6
SCHEMBL7019824 0.86 CA12 (0.65) CA12CA1CA2CA4CA6
SCHEMBL30221732 0.86 CA12 (0.65) CA12CA1CA2CA4CA6
SCHEMBL129159 0.86 HDAC1 (0.57) HTTLMNAALDH1A1MAPTKDM4E
SCHEMBL310059 0.86 MAPT (0.60) CA12CA1CA2CA4CA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117658749-B Method for preparing aryl carboxylic acid by reacting copper compound catalyzed aryl sulfonium salt with carbon dioxide NANKAI UNIVERSITY (CN) 2026-05-26 CN disclosed
EP-4448508-A1 BENZOTHIOPHENE DERIVATIVES AS RXFP1 AGONISTS Bristol-Myers Squibb Company (US) 2024-10-23 EP disclosed
CN-118647606-A Benzothiophene derivatives as RXFP1 agonists 百时美施贵宝公司 2024-09-13 CN disclosed
CN-118401502-A Benzothiazole, benzisoxazole and benzodioxole analogs as RXFP1 receptor agonists 百时美施贵宝公司 2024-07-26 CN disclosed
CN-117658749-A Method for preparing aryl carboxylic acid by reacting copper compound catalyzed aryl sulfonium salt with carbon dioxide 南开大学 2024-03-08 CN disclosed
CN-111295382-B Bridged bicyclic compounds as farnesyl ester X receptor modulators 百时美施贵宝公司 2024-02-02 CN disclosed
CN-117024319-A Amide compound, pharmaceutical composition containing same, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2023-11-10 CN disclosed
CN-110724075-B Amide compound, pharmaceutical composition containing same, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2023-09-12 CN disclosed
WO-2023114823-A1 BENZOTHIOPHENE DERIVATIVES AS RXFP1 AGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2023-06-22 WO disclosed