SCHEMBL30457738

SCHEMBL30457738

COC(=O)c1cc(N)c2sc(C(F)(F)F)nc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.40
ALDH1A1 P00352 4/20 0.40
NOTUM Q6P988 2/20 0.40
LMNA P02545 2/20 0.40
HTT P42858 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MAPT P10636 5/20 0.39
HPGD P15428 3/20 0.39
GAA P10253 2/20 0.39
GLA P06280 1/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
ATM Q13315 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CFTR P13569 3/20 0.39
KMT2A Q03164 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
MEN1 O00255 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25284930 1.00 KDM4E (0.40) KDM4EALDH1A1NOTUMLMNAHTT
SCHEMBL30458112 0.76 HTT (0.50) KDM4EALDH1A1NOTUMLMNAHTT
SCHEMBL25234075 0.76 HTT (0.50) KDM4EALDH1A1NOTUMLMNAHTT
SCHEMBL25233286 0.74 CFTR (0.49) KDM4EALDH1A1MAPTHPGDGAA
SCHEMBL30457719 0.74 CFTR (0.49) KDM4EALDH1A1MAPTHPGDGAA
SCHEMBL20839800 0.69 MAPT (0.46) KDM4EALDH1A1NOTUML3MBTL1MAPT
SCHEMBL27901095 0.68 NOTUM (0.51) KDM4EALDH1A1NOTUMLMNAL3MBTL1
SCHEMBL23826015 0.67 NOTUM (0.46) KDM4EALDH1A1NOTUMLMNAL3MBTL1
SCHEMBL30152983 0.67 CFTR (0.50) KDM4EALDH1A1NOTUMLMNAL3MBTL1
SCHEMBL753404 0.67 CFTR (0.50) KDM4EALDH1A1NOTUMLMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4448500-A1 BENZOTHIAZOLE, BENZOISOXAZOLE AND BENZODIOXOLE ANALOGS AS RXFP1 RECEPTOR AGONISTS Bristol-Myers Squibb Company (US) 2024-10-23 EP disclosed
WO-2023114822-A1 BENZOTHIAZOLE, BENZOISOXAZOLE AND BENZODIOXOLE ANALOGS AS RXFP1 RECEPTOR AGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2023-06-22 WO disclosed