SCHEMBL30458549

SCHEMBL30458549

CC(=O)Nc1ccn(C(=O)N2CCC3(CCN(Cc4cc(C(F)(F)F)cc(C5(C(=O)O)CCCC5)c4)C3)CC2)n1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
FAAH O00519 6/20 0.57
MGLL Q99685 2/20 0.49
CYP3A4 P08684 9/20 0.49
CYP2D6 P10635 7/20 0.49
TSHR P16473 6/20 0.49
ALDH1A1 P00352 1/20 0.47
USP2 O75604 7/20 0.45
HPGD P15428 1/20 0.45
CYP2C19 P33261 2/20 0.44
CYP1A2 P05177 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
HIF1A Q16665 2/20 0.43
CYP2C9 P11712 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20570710 1.00 FAAH (0.57) FAAHMGLLCYP3A4CYP2D6TSHR
SCHEMBL20571312 0.91 FAAH (0.52) FAAHMGLLCYP3A4CYP2D6TSHR
SCHEMBL31168842 0.91 FAAH (0.52) FAAHMGLLCYP3A4CYP2D6TSHR
SCHEMBL21896123 0.86 FAAH (0.53) FAAHMGLLCYP3A4CYP2D6TSHR
SCHEMBL21896151 0.84 FAAH (0.57) FAAHMGLLCYP3A4CYP2D6TSHR
SCHEMBL21896137 0.84 MGLL (0.46) FAAHMGLL
SCHEMBL21821118 0.82 FAAH (0.43) FAAHMGLL
SCHEMBL31168819 0.82 FAAH (0.43) FAAHMGLL
SCHEMBL21821182 0.77 FAAH (0.62) FAAHMGLL
SCHEMBL31168783 0.77 FAAH (0.62) FAAHMGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110678177-B Pyrazole MAGL inhibitors H.隆德贝克有限公司 2023-06-13 CN disclosed