SCHEMBL30459933

SCHEMBL30459933

COc1ccc(Nc2ccnc(Cl)n2)c([N+](=O)[O-])c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 4/20 0.50
AKR1C2 P52895 4/20 0.50
KCNMA1 Q12791 1/20 0.48
MAPT P10636 6/20 0.48
MAPK1 P28482 2/20 0.48
ALDH1A1 P00352 2/20 0.48
TDP1 Q9NUW8 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
AKR1B10 O60218 1/20 0.47
AKR1B1 P15121 1/20 0.47
AKR1C4 P17516 1/20 0.47
AKR1C1 Q04828 1/20 0.47
PIN1 Q13526 1/20 0.46
NPC1 O15118 5/20 0.46
RAB9A P51151 4/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C19 P33261 1/20 0.46
SMN1; SMN2 Q16637 4/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17683159 1.00 AKR1C3 (0.50) AKR1C3AKR1C2KCNMA1MAPTMAPK1
SCHEMBL30108026 0.84 AKR1C3 (0.51) AKR1C3AKR1C2KCNMA1MAPTMAPK1
SCHEMBL30724421 0.84 AKR1C3 (0.48) AKR1C3AKR1C2KCNMA1MAPTMAPK1
SCHEMBL21642825 0.84 AKR1C3 (0.48) AKR1C3AKR1C2KCNMA1MAPTMAPK1
SCHEMBL6176751 0.80 GAA (0.59) AKR1C3AKR1C2KCNMA1MAPTMAPK1
SCHEMBL4820325 0.80 GAA (0.62) MAPTMAPK1ALDH1A1L3MBTL1NPC1
SCHEMBL31220866 0.79 MEN1 (0.68) AKR1C3AKR1C2KCNMA1MAPTMAPK1
SCHEMBL17683162 0.79 ROCK1 (0.47) MAPTMAPK1ALDH1A1L3MBTL1NPC1
SCHEMBL30459783 0.79 ROCK1 (0.47) MAPTMAPK1ALDH1A1L3MBTL1NPC1
SCHEMBL3638254 0.77 LCK (0.56) MAPTMAPK1ALDH1A1L3MBTL1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117402143-A EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2024-01-16 CN disclosed
CN-117069700-A EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-11-17 CN disclosed
CN-111187221-B EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-09-26 CN disclosed
CN-111171000-B EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-09-01 CN disclosed
CN-111170999-B EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-06-30 CN disclosed