SCHEMBL30462004

SCHEMBL30462004

FC(F)(F)c1ccc(-c2ccc(CCl)cc2)nc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.51
CYP11B1 P15538 1/20 0.46
CYP11B2 P19099 1/20 0.46
MAOB P27338 2/20 0.46
KDM1A O60341 2/20 0.46
PPARA Q07869 2/20 0.42
P2RX7 Q99572 1/20 0.40
NPSR1 Q6W5P4 2/20 0.40
LTA4H P09960 1/20 0.40
KDM4E B2RXH2 1/20 0.39
EPHB4 P54760 2/20 0.39
GCK P35557 1/20 0.39
GCKR Q14397 1/20 0.39
TEK Q02763 2/20 0.38
KDR P35968 1/20 0.38
MCHR1 Q99705 1/20 0.37
PPARD Q03181 1/20 0.37
HDAC1 Q13547 1/20 0.37
KMT2A Q03164 1/20 0.37
CASP3 P42574 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3387516 1.00 KIF11 (0.51) KIF11CYP11B1CYP11B2MAOBKDM1A
Hydrochloric Acid SCHEMBL31453978 0.98 KIF11 (0.50) KIF11CYP11B1CYP11B2MAOBKDM1A
SCHEMBL1550000 0.90 CYP11B1 (0.49) KIF11CYP11B1CYP11B2MAOBKDM1A
Hydrochloric Acid SCHEMBL31375590 0.89 CYP11B1 (0.48) KIF11CYP11B1CYP11B2MAOBKDM1A
SCHEMBL30767444 0.87 KIF11 (0.40) KIF11CYP11B1CYP11B2MAOBKDM1A
SCHEMBL27344645 0.86 KIF11 (0.63) KIF11CYP11B1CYP11B2MAOBKDM1A
SCHEMBL14037163 0.85 KIF11 (0.52) KIF11CYP11B1CYP11B2MAOBKDM1A
SCHEMBL29690424 0.84 KIF11 (0.61) KIF11CYP11B1CYP11B2MAOBKDM1A
SCHEMBL28530523 0.84 KIF11 (0.61) KIF11CYP11B1CYP11B2MAOBKDM1A
SCHEMBL8239616 0.83 KIF11 (0.51) KIF11CYP11B1CYP11B2MAOBKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4568959-A1 BICYCLIC TETRAHYDROTHIAZEPINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2025-06-18 EP disclosed
CN-119677733-A Bicyclic tetrahydrothiazepine derivatives 豪夫迈·罗氏有限公司 2025-03-21 CN disclosed
CN-118660872-A Pyrimidine compound, preparation method and medical application thereof 江苏亚虹医药科技股份有限公司 2024-09-17 CN disclosed
CN-116496252-A Pyrimidine compound, preparation method and medical application thereof 江苏亚虹医药科技股份有限公司 2023-07-28 CN disclosed