SCHEMBL30463555

SCHEMBL30463555

Nc1coc(-c2ccco2)c1-c1ccncn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 16/20 0.46
ADORA1 P30542 12/20 0.46
ADORA2A P29274 10/20 0.46
MAPK1 P28482 2/20 0.45
TDP1 Q9NUW8 2/20 0.45
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
ALDH1A1 P00352 1/20 0.45
POLB P06746 1/20 0.45
MAPT P10636 1/20 0.45
THRB P10828 1/20 0.45
PKM P14618 1/20 0.45
HPGD P15428 1/20 0.45
ALOX15 P16050 1/20 0.45
APEX1 P27695 1/20 0.45
BRCA1 P38398 1/20 0.45
RECQL P46063 1/20 0.45
BLM P54132 1/20 0.45
CASP7 P55210 1/20 0.45
CACNA1B Q00975 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1445253 0.79 MAPK1 (0.53) ADORA2BADORA1ADORA2AMAPK1KDM4E
SCHEMBL30463614 0.79 MAPK1 (0.53) ADORA2BADORA1ADORA2AMAPK1KDM4E
SCHEMBL3061780 0.73 ADORA2B (0.54) ADORA2BADORA1ADORA2ATDP1KDM4E
SCHEMBL4057562 0.73 ADORA2B (0.61) ADORA2BADORA1ADORA2AADORA3MAP4K4
SCHEMBL28758987 0.73 ADORA2B (0.51) ADORA2BADORA1ADORA2AMAPK1TDP1
SCHEMBL28135936 0.72 ADORA2B (0.53) ADORA2BADORA1ADORA2AKDM4EALDH1A1
SCHEMBL4049097 0.71 ADORA2B (0.64) ADORA2BADORA1ADORA2AADORA3MAP4K4
SCHEMBL3058599 0.70 ADORA2B (0.57) ADORA2BADORA1ADORA2ATDP1KDM4E
SCHEMBL29769313 0.70 TAAR1 (0.45) ADORA1ADORA2AMAPK1TDP1KDM4E
SCHEMBL4052108 0.70 ADORA2B (0.61) ADORA2BADORA1ADORA2AADORA3MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116514799-A Wee1 inhibitor, composition and application thereof 星希尔生物科技(上海)有限公司 2023-08-01 CN disclosed