SCHEMBL30468397

SCHEMBL30468397

COc1ccc2c(c1)CC(=O)NC=C2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 1.00
METAP1 P53582 2/20 0.43
PDE3B Q13370 3/20 0.41
PDE3A Q14432 3/20 0.41
SRC P12931 2/20 0.39
TDP2 O95551 1/20 0.39
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
MAOB P27338 3/20 0.38
MAOA P21397 2/20 0.38
ALDH1A1 P00352 1/20 0.37
DRD2 P14416 1/20 0.37
DRD1 P21728 1/20 0.37
DRD5 P21918 1/20 0.37
DRD3 P35462 1/20 0.37
BCL2 P10415 1/20 0.36
ACHE P22303 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL227653 1.00 GAA (1.00) GAAMETAP1PDE3BPDE3ASRC
SCHEMBL11044464 0.81 GAA (0.68) GAAMETAP1PDE3BPDE3ACYP11B1
SCHEMBL333847 0.78 GAA (0.63) GAASRCMAOAALDH1A1ACHE
SCHEMBL5044573 0.76 GAA (0.60) GAAPDE3BPDE3ATDP2MAOB
SCHEMBL21762103 0.74 GAA (0.58) GAAMETAP1PDE3BPDE3ASRC
SCHEMBL28634068 0.74 GAA (0.58) GAASRCTDP2
SCHEMBL19038489 0.73 GAA (0.58) GAAMETAP1PDE3BPDE3ACYP11B1
SCHEMBL10232028 0.73 GAA (0.57) GAAMETAP1PDE3BPDE3ACYP11B1
SCHEMBL15906664 0.73 GAA (0.57) GAAMAOAALDH1A1ACHE
SCHEMBL11045652 0.73 GAA (0.57) GAATDP2ALDH1A1DRD5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115594669-B Parallel ring derivative and preparation method and medical application thereof 深圳信立泰药业股份有限公司 2024-11-05 CN disclosed
CN-116332910-A 2-aminopyrimidine derivatives as kinase inhibitors, preparation and use thereof 江苏威凯尔医药科技有限公司 2023-06-27 CN disclosed