SCHEMBL11045652

SCHEMBL11045652

COc1cc2c(cc1F)CC(=O)NC=C2

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.57
BRD4 O60885 1/20 0.44
TDP2 O95551 2/20 0.41
NCOA1 Q15788 1/20 0.36
NCOA3 Q9Y6Q9 1/20 0.36
HTR1A P08908 1/20 0.32
CYP3A4 P08684 1/20 0.32
MAPT P10636 1/20 0.32
HTR2B P41595 1/20 0.32
TIPARP Q7Z3E1 1/20 0.31
MTNR1A P48039 1/20 0.31
MTNR1B P49286 1/20 0.31
DRD5 P21918 1/20 0.31
CRHBP P24387 1/20 0.31
CRHR2 Q13324 1/20 0.31
LMNA P02545 1/20 0.30
MAPK1 P28482 1/20 0.30
HTT P42858 1/20 0.30
RAB9A P51151 1/20 0.30
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL333847 0.88 GAA (0.63) GAABRD4CYP3A4MAPTCRHBP
SCHEMBL11041542 0.82 BRD4 (0.38) GAABRD4TDP2NCOA1NCOA3
SCHEMBL15906664 0.82 GAA (0.57) GAABRD4ALDH1A1
Oxalic Acid SCHEMBL15319252 0.81 GAA (0.56) GAABRD4CYP3A4MAPTCRHBP
SCHEMBL28634068 0.81 GAA (0.58) GAABRD4TDP2CYP3A4MAPT
SCHEMBL13593675 0.76 GAA (0.53) GAABRD4CYP3A4MAPTCRHBP
SCHEMBL3821050 0.75 PARP1 (0.37) BRD4TDP2NCOA1NCOA3CYP3A4
SCHEMBL11041593 0.75 GAA (0.51) GAABRD4CYP3A4MAPTMAPK1
SCHEMBL11043204 0.73 BRD4 (0.44) BRD4TDP2NCOA1NCOA3CYP3A4
SCHEMBL30468397 0.73 GAA (1.00) GAATDP2DRD5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0116444-A2 Improvements in or relating to benzazepine derivatives ELI LILLY AND COMPANY (US) 1984-08-22 EP disclosed