SCHEMBL3047451

SCHEMBL3047451

COc1cccc(S(=O)(=O)Oc2ccc(-c3cc4cc(CN5CCCCC5)ccc4n3C(=O)OC(C)(C)C)c3c2CNC3=O)c1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 9/20 0.40
CNR2 P34972 1/20 0.35
ATR Q13535 1/20 0.34
ATRIP Q8WXE1 1/20 0.34
ROCK2 O75116 1/20 0.34
CCR2 P41597 1/20 0.33
HTR6 P50406 1/20 0.33
POLB P06746 1/20 0.33
TGFBR1 P36897 1/20 0.32
MCHR1 Q99705 1/20 0.32
ACHE P22303 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3054403 0.93 NR1H2 (0.36) NR1H2CNR2ATRATRIPPOLB
SCHEMBL3039560 0.92 NR1H2 (0.40) NR1H2
SCHEMBL3047662 0.92 NR1H2 (0.37) NR1H2CCR2
SCHEMBL3049978 0.92 NR1H2 (0.39) NR1H2
SCHEMBL3045896 0.92 MEN1 (0.34) NR1H2ACHE
SCHEMBL3047368 0.90 HTR6 (0.38) NR1H2HTR6
SCHEMBL3048398 0.90 NR1H2 (0.36) NR1H2ATRATRIPACHE
SCHEMBL3044144 0.89 NR1H2 (0.33) NR1H2ATRATRIP
SCHEMBL3040219 0.89 NR1H2 (0.34) NR1H2HTR6
SCHEMBL3042182 0.89 NR1H2 (0.40) NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7745641-B2 Nitrogen-containing heterocyclic compound KYOWA HAKKO KIRIN CO., LTD. (JP) 2010-06-29 US disclosed
US-20090054407-A1 Nitrogen-containing heterocyclic compound KYOWA HAKKO KOGYO CO., LTD. (JP) 2009-02-26 US disclosed
EP-1880993-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND KYOWA HAKKO KOGYO CO., LTD. (JP) 2008-01-23 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090054407-A1 Nitrogen-containing heterocyclic compound NR4A1, NR5A2, PRMT8 NR1H2 21/4885CNR2 134/4885ATR 1385/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.