SCHEMBL30476247

SCHEMBL30476247

CN1C(=O)COc2ccc(Br)c(F)c21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.38
HTR1D P28221 2/20 0.38
HTR1B P28222 2/20 0.38
PDE3B Q13370 2/20 0.38
PDE3A Q14432 2/20 0.38
BRD4 O60885 2/20 0.35
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
TSHR P16473 1/20 0.33
HTT P42858 1/20 0.33
GPR55 Q9Y2T6 1/20 0.33
GRM4 Q14833 1/20 0.32
KMO O15229 1/20 0.32
PLK1 P53350 1/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.31
TERT O14746 1/20 0.31
GABRG2 P18507 1/20 0.30
GABRB3 P28472 1/20 0.30
GABRA5 P31644 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4170716 0.76 HTR1A (0.43) HTR1AHTR1DHTR1BPDE3BPDE3A
SCHEMBL31180323 0.75 PDE3B (0.37) HTR1AHTR1DHTR1BPDE3BPDE3A
SCHEMBL30336343 0.74 TERT (0.41) HTR1AHTR1DHTR1BPDE3BPDE3A
SCHEMBL16738955 0.74 BRD4 (0.56) HTR1AHTR1DHTR1BPDE3BPDE3A
SCHEMBL30336272 0.72 PDE3B (0.35) PDE3BPDE3ACYP11B1CYP11B2TSHR
SCHEMBL29209037 0.72 PDE3B (0.35) PDE3BPDE3ACYP11B1CYP11B2TSHR
Hydrochloric Acid SCHEMBL6831442 0.69 HTR1A (0.41) HTR1AHTR1DHTR1BPDE3BPDE3A
SCHEMBL10442160 0.69 HTR1A (0.42) HTR1AHTR1DHTR1BPDE3BPDE3A
SCHEMBL11572747 0.69 MEN1 (0.42) HTR1AHTR1DHTR1BPDE3BPDE3A
SCHEMBL29209156 0.69 PDE3B (0.43) HTR1APDE3BPDE3ACYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116332937-A Dipeptidyl peptidase I inhibitors and uses thereof 杭州邦顺制药有限公司 2023-06-27 CN disclosed