SCHEMBL30480717

SCHEMBL30480717

CC1(C)COB(c2ccc(C#N)cc2N)O1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
NSD2 O96028 1/20 0.33
PDE4B Q07343 3/20 0.32
PDE4A P27815 2/20 0.32
PDE4C Q08493 2/20 0.32
PDE4D Q08499 2/20 0.32
MALT1 Q9UDY8 1/20 0.32
CHRM1 P11229 1/20 0.31
ADRA1A P35348 1/20 0.31
PDE1A P54750 1/20 0.31
PDE3B Q13370 1/20 0.31
PDE7A Q13946 1/20 0.31
PDE3A Q14432 1/20 0.31
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL614874 0.86 KDM4E (0.37) KDM4EALDH1A1GAANSD2PDE4B
SCHEMBL12069815 0.83 AR (0.33) PDE4BPDE4APDE4CPDE4DMALT1
SCHEMBL22637023 0.81 ALDH1A1 (0.36) KDM4EALDH1A1GAANSD2PDE4B
SCHEMBL30372881 0.81 ALDH1A1 (0.36) KDM4EALDH1A1GAANSD2PDE4B
SCHEMBL28967143 0.80 MALT1 (0.30) PDE4BMALT1
SCHEMBL29053479 0.78 ALDH1A1 (0.35) ALDH1A1GAAPDE3A
SCHEMBL23422357 0.77 NSD2 (0.37) NSD2PDE4BPDE4APDE4CPDE4D
SCHEMBL31448668 0.71 TSHR (0.35) PDE4BPDE4APDE4CPDE4D
SCHEMBL16924038 0.70 ALDH1A1 (0.34) KDM4EALDH1A1GAANSD2MALT1
SCHEMBL20920749 0.69 AR (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107973809-B Macrocyclic compounds as factor XIA inhibitors 百时美施贵宝公司 2023-06-30 CN disclosed