SCHEMBL30482190

SCHEMBL30482190

Cc1cccc(CN(Cc2ccccn2)C(=O)C(N)=O)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RECQL P46063 3/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C9 P11712 1/20 0.54
CYP2C19 P33261 1/20 0.54
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.46
TSHR P16473 2/20 0.45
ALDH1A1 P00352 2/20 0.45
NPSR1 Q6W5P4 2/20 0.45
TRPM8 Q7Z2W7 1/20 0.45
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
KDM4E B2RXH2 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 2/20 0.42
NR3C2 P08235 1/20 0.42
VNN1 O95497 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25373830 1.00 RECQL (0.54) RECQLCYP2D6CYP2C9CYP2C19MEN1
SCHEMBL25373467 0.92 RECQL (0.47) RECQLCYP2D6CYP2C9CYP2C19MEN1
SCHEMBL25375508 0.86 MEN1 (0.58) RECQLMEN1KMT2AL3MBTL1TSHR
SCHEMBL25375460 0.86 L3MBTL1 (0.60) RECQLMEN1KMT2AL3MBTL1TSHR
SCHEMBL30482189 0.85 RECQL (0.51) RECQLCYP2D6CYP2C9CYP2C19MEN1
SCHEMBL25377248 0.85 RECQL (0.51) RECQLCYP2D6CYP2C9CYP2C19MEN1
SCHEMBL25377677 0.84 SMN1; SMN2 (0.50) MEN1KMT2AL3MBTL1TSHRALDH1A1
SCHEMBL25378936 0.84 L3MBTL1 (0.46) MEN1KMT2AL3MBTL1TSHRALDH1A1
SCHEMBL25375114 0.79 KDM4E (0.54) MEN1KMT2AL3MBTL1TSHRALDH1A1
SCHEMBL25376675 0.78 TRPM8 (0.54) RECQLMEN1KMT2AL3MBTL1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4469438-A1 COMPOUNDS AND METHODS OF USE Tango Therapeutics, Inc. (US) 2024-12-04 EP disclosed
WO-2023146987-A1 COMPOUNDS AND METHODS OF USE TANGO THERAPEUTICS, INC. (US) 2023-08-03 WO disclosed