SCHEMBL30482452

SCHEMBL30482452

Fc1cccnc1-c1cncs1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 3/20 0.45
DYRK1A Q13627 2/20 0.41
DYRK2 Q92630 1/20 0.41
DYRK1B Q9Y463 1/20 0.41
CD38 P28907 3/20 0.39
GABRG2 P18507 7/20 0.38
GABRB3 P28472 7/20 0.38
GABRA5 P31644 7/20 0.38
GABRA3 P34903 7/20 0.38
GABRA1 P14867 6/20 0.38
ADORA3 P0DMS8 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA2B P29275 1/20 0.38
ADORA1 P30542 1/20 0.38
TBXAS1 P24557 1/20 0.38
HDAC4 P56524 1/20 0.37
LRRK2 Q5S007 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27164862 1.00 PIM1 (0.45) PIM1DYRK1ADYRK2DYRK1BCD38
SCHEMBL24568619 0.79 CYP2A6 (0.51) PIM1DYRK1ADYRK2DYRK1BCD38
SCHEMBL24567811 0.75 TBXAS1 (0.41) PIM1DYRK1ADYRK2DYRK1BCD38
SCHEMBL7430359 0.74 CYP11B1 (0.47) ADORA2A
SCHEMBL5088040 0.73 KDM4E (0.61) PIM1DYRK1ADYRK2DYRK1BTBXAS1
SCHEMBL15624391 0.73 TDP1 (0.44) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL28273959 0.73 HDAC4 (0.43) PIM1DYRK1ADYRK2DYRK1BCD38
SCHEMBL28416665 0.73 PIM1 (0.41) PIM1DYRK1ADYRK2DYRK1BCD38
SCHEMBL15638356 0.73 CD38 (0.46) PIM1DYRK1ADYRK2DYRK1BCD38
SCHEMBL19302641 0.72 PIM1 (0.51) PIM1DYRK1ADYRK2DYRK1BCD38

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4469035-A1 IMIDAZOPYRIDINE INHIBITORS OF TYROSINE KINASE Bridgene Biosciences, Inc. (US) 2024-12-04 EP disclosed
WO-2023146786-A1 IMIDAZOPYRIDINE INHIBITORS OF TYROSINE KINASE BRIDGENE BIOSCIENCES, INC. (US) 2023-08-03 WO disclosed