SCHEMBL30484456

SCHEMBL30484456

c1ccc(-c2ccc(-c3ccnc(CN4CCC5(CC4)OCCc4ccsc45)c3)cc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.52
OPRL1 P41146 6/20 0.48
SIGMAR1 Q99720 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29204480 0.85 SIGMAR1 (0.61) SIGMAR1
SCHEMBL30484429 0.78 EGLN1 (0.46) OPRL1SIGMAR1
SCHEMBL30484402 0.76 SIGMAR1 (0.56) RORCOPRL1SIGMAR1
SCHEMBL30484446 0.75 EGLN1 (0.43) OPRL1SIGMAR1
SCHEMBL29204466 0.74 EGLN1 (0.48) OPRL1SIGMAR1
SCHEMBL29204460 0.74 EGLN1 (0.48) OPRL1SIGMAR1
SCHEMBL30484462 0.73 EGLN1 (0.47) OPRL1SIGMAR1
SCHEMBL29204511 0.72 EGLN1 (0.46) OPRL1SIGMAR1
SCHEMBL10374628 0.72 OPRL1 (0.56) OPRL1SIGMAR1
SCHEMBL30484482 0.72 EGLN1 (0.46) OPRL1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116354897-B Substituted 1,2, 4-triazole, pyridine and pyrimidine derivatives and application thereof in medicines 华东师范大学 2024-10-15 CN disclosed
CN-116354897-A Substituted 1,2, 4-triazole, pyridine and pyrimidine derivatives and application thereof in medicines 华东师范大学 2023-06-30 CN disclosed