SCHEMBL30484402

SCHEMBL30484402

Cn1nc(CN2CCC3(CC2)OCCc2ccsc23)nc1-c1ccc(-c2ccccc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.56
TMEM97 Q5BJF2 3/20 0.48
RORC P51449 1/20 0.48
OPRL1 P41146 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29204513 0.89 SIGMAR1 (0.58) SIGMAR1TMEM97RORCOPRL1
SCHEMBL29204508 0.89 SIGMAR1 (0.58) SIGMAR1TMEM97RORC
SCHEMBL29204493 0.86 SIGMAR1 (0.59) SIGMAR1TMEM97
SCHEMBL29204426 0.77 SIGMAR1 (0.59) SIGMAR1TMEM97
SCHEMBL29204462 0.77 SIGMAR1 (0.59) SIGMAR1TMEM97
SCHEMBL30484456 0.76 RORC (0.52) SIGMAR1RORCOPRL1
SCHEMBL29204475 0.75 RORC (0.44) SIGMAR1TMEM97RORCOPRL1
SCHEMBL31252997 0.75 SIGMAR1 (0.41) SIGMAR1TMEM97OPRL1
SCHEMBL30056578 0.74 SIGMAR1 (1.00) SIGMAR1TMEM97
SCHEMBL11949323 0.71 RORC (0.55) SIGMAR1RORCOPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116354897-B Substituted 1,2, 4-triazole, pyridine and pyrimidine derivatives and application thereof in medicines 华东师范大学 2024-10-15 CN disclosed
CN-116354897-A Substituted 1,2, 4-triazole, pyridine and pyrimidine derivatives and application thereof in medicines 华东师范大学 2023-06-30 CN disclosed