SCHEMBL30495014

SCHEMBL30495014

Cc1cc(Br)c2nc(-c3cccc(F)c3)n(C)c(=O)c2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.39
ADORA2B P29275 5/20 0.39
ADORA1 P30542 5/20 0.39
ADORA3 P0DMS8 4/20 0.39
ALDH1A1 P00352 3/20 0.39
USP2 O75604 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
TSHR P16473 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
PTGS2 P35354 2/20 0.38
PTGS1 P23219 1/20 0.38
KDM4E B2RXH2 2/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
BACE1 P56817 1/20 0.37
TNKS2 Q9H2K2 1/20 0.37
TP53 P04637 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25360538 1.00 ADORA2A (0.39) ADORA2AADORA2BADORA1ADORA3ALDH1A1
SCHEMBL25361244 0.86 KDM4E (0.38) ADORA2AADORA1ADORA3CYP3A4KDM4E
SCHEMBL30858003 0.86 KDM4E (0.38) ADORA2AADORA1ADORA3CYP3A4KDM4E
SCHEMBL30494909 0.86 ADORA2B (0.43) ADORA2AADORA2BADORA1ADORA3ALDH1A1
SCHEMBL25359782 0.86 ADORA2B (0.43) ADORA2AADORA2BADORA1ADORA3ALDH1A1
SCHEMBL30690334 0.82 EGFR (0.37)
SCHEMBL25360145 0.82 DHODH (0.41) ADORA2AADORA2BADORA1ADORA3ALDH1A1
SCHEMBL25360382 0.81 ADORA2A (0.39) ADORA2AADORA2BADORA1ADORA3ALDH1A1
SCHEMBL25360386 0.81 ADORA2A (0.39) ADORA2AADORA2BADORA1ADORA3ALDH1A1
SCHEMBL30495001 0.81 ADORA2A (0.39) ADORA2AADORA2BADORA1ADORA3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023159155-A1 INHIBITORS OF PHOSPHOINOSITIDE 3-KINASE (PI3K) AND USES THEREOF PIVALENT THERAPEUTICS, INC. (US) 2023-08-24 WO disclosed