SCHEMBL30690334

SCHEMBL30690334

Cc1cc(Br)c2nc(-c3c(F)cccc3F)n(C)c(=O)c2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.37
JAK2 O60674 1/20 0.37
BTK Q06187 1/20 0.37
ADRA1A P35348 1/20 0.35
KCNH2 Q12809 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
DHODH Q02127 2/20 0.35
PDE2A O00408 1/20 0.34
PDE10A Q9Y233 1/20 0.34
PKM P14618 2/20 0.34
PTGES O14684 3/20 0.33
WEE1 P30291 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
PDE7A Q13946 1/20 0.33
PDE7B Q9NP56 1/20 0.33
AADAT Q8N5Z0 1/20 0.33
CYP2D6 P10635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30495148 0.86 HSD11B1 (0.40) EGFRDHODHPTGES
SCHEMBL25358826 0.86 HSD11B1 (0.40) EGFRDHODHPTGES
SCHEMBL26042227 0.84 DHODH (0.37) ADRA1AKCNH2HRH3DHODHPTGES
SCHEMBL30495014 0.82 ADORA2A (0.39)
SCHEMBL25360538 0.82 ADORA2A (0.39)
SCHEMBL30690320 0.81 DHODH (0.42) ADRA1AKCNH2HRH3DHODHPTGES
SCHEMBL29139168 0.81 AKT1 (0.35) ADRA1AKCNH2HRH3DHODHPTGES
SCHEMBL30690342 0.81 AKT1 (0.35) ADRA1AKCNH2HRH3DHODHPTGES
SCHEMBL29139165 0.81 AKT1 (0.35) ADRA1AKCNH2HRH3DHODHPTGES
SCHEMBL25361244 0.81 KDM4E (0.38) EGFRADRA1AKCNH2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117362281-A PI3K inhibitor and preparation method and application thereof 海创药业股份有限公司 2024-01-09 CN disclosed