SCHEMBL30499545

SCHEMBL30499545

CC(C)C(=O)N1CC=C(c2cc(-c3ccc(NC(=O)OC(C)(C)C)cc3)c3c(N)ncnc3c2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.49
NAMPT P43490 11/20 0.45
BTK Q06187 1/20 0.41
HCK P08631 2/20 0.41
SRC P12931 2/20 0.41
LCK P06239 1/20 0.41
FYN P06241 1/20 0.41
LYN P07948 1/20 0.41
FRK P42685 1/20 0.41
BLK P51451 1/20 0.41
PTK6 Q13882 1/20 0.41
KIT P10721 1/20 0.39
PIK3CD O00329 2/20 0.39
ABL1 P00519 2/20 0.39
EGFR P00533 2/20 0.39
KDR P35968 2/20 0.39
PIK3CA P42336 2/20 0.39
PIK3CG P48736 2/20 0.39
PRKDC P78527 2/20 0.39
PIK3CB P42338 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29052739 1.00 MAP4K4 (0.49) MAP4K4NAMPTBTKHCKSRC
SCHEMBL29052499 0.82 NAMPT (0.40) MAP4K4NAMPTBTKLCKKIT
SCHEMBL29052482 0.82 MAP4K4 (0.49) MAP4K4NAMPTHCKSRCLCK
SCHEMBL30499549 0.82 MAP4K4 (0.49) MAP4K4NAMPTHCKSRCLCK
SCHEMBL30499541 0.76 MAP4K4 (0.62) MAP4K4HCKSRCLCKFYN
SCHEMBL29052462 0.76 MAP4K4 (0.62) MAP4K4HCKSRCLCKFYN
SCHEMBL30367031 0.68 NAMPT (0.43) MAP4K4NAMPTLCKLYNFRK
SCHEMBL22418461 0.68 FLT3 (0.62) MAP4K4HCKSRCLCKFYN
SCHEMBL24891722 0.67 NAMPT (0.63) NAMPTKITCDK7CDK13CDK12
SCHEMBL15587426 0.67 MAP4K4 (1.00) MAP4K4HCKSRCPIK3CDABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116437918-A Pyrazolopyridine compounds as TAM inhibitors 上海德琪医药科技有限公司 2023-07-14 CN disclosed