SCHEMBL30508265

SCHEMBL30508265

COC(=O)c1cc(-c2ccc(CN3CCOCC3)cc2)cnc1N

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AXL P30530 4/20 0.58
MERTK Q12866 4/20 0.58
TBK1 Q9UHD2 6/20 0.55
LRRK2 Q5S007 2/20 0.52
IKBKE Q14164 5/20 0.51
ACVR1 Q04771 3/20 0.50
BMPR1B O00238 2/20 0.50
BMPR1A P36894 2/20 0.50
TGFBR1 P36897 2/20 0.50
ACVRL1 P37023 2/20 0.50
MAP4K1 Q92918 1/20 0.49
MAPK1 P28482 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
HRH3 Q9Y5N1 1/20 0.49
HCRTR1 O43613 1/20 0.48
HCRTR2 O43614 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29042029 1.00 AXL (0.58) AXLMERTKTBK1LRRK2IKBKE
SCHEMBL30508238 0.87 LRRK2 (0.57) AXLMERTKTBK1LRRK2IKBKE
SCHEMBL18611468 0.87 AXL (0.55) AXLMERTKTBK1LRRK2IKBKE
SCHEMBL30508270 0.86 LRRK2 (0.56) AXLMERTKLRRK2MAP4K1MAPK1
SCHEMBL29041987 0.86 LRRK2 (0.56) AXLMERTKLRRK2MAP4K1MAPK1
SCHEMBL30508414 0.85 BMPR1B (0.64) TBK1IKBKEACVR1BMPR1BBMPR1A
SCHEMBL29152375 0.85 BMPR1B (0.64) TBK1IKBKEACVR1BMPR1BBMPR1A
SCHEMBL31027897 0.82 SMN1; SMN2 (0.50) AXLMERTKMAPK1SMN1; SMN2HRH3
SCHEMBL4126100 0.82 MAP4K1 (0.65) AXLMAP4K1
SCHEMBL29041913 0.82 ACVR1 (0.67) AXLMERTKACVR1BMPR1BBMPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116478145-B ALK2 kinase inhibitors 杭州邦顺制药有限公司 2024-02-02 CN disclosed
CN-116478145-A ALK2 kinase inhibitors 杭州邦顺制药有限公司 2023-07-25 CN disclosed