SCHEMBL30508288

SCHEMBL30508288

COC(=O)c1cc(-c2ccc3nn(C4CCN(C5COC5)CC4)cc3c2)cnc1N

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 4/20 0.45
GSK3B P49841 3/20 0.42
DYRK1A Q13627 3/20 0.42
WNT1 P04628 2/20 0.42
BMPR1B O00238 4/20 0.40
BMPR1A P36894 4/20 0.40
TGFBR1 P36897 4/20 0.40
ACVRL1 P37023 4/20 0.40
ACVR1 Q04771 4/20 0.40
MET P08581 2/20 0.39
MAP3K12 Q12852 3/20 0.38
TLR8 Q9NR97 1/20 0.38
IKBKE Q14164 1/20 0.37
TBK1 Q9UHD2 1/20 0.37
MAP4K3 Q8IVH8 1/20 0.37
AXL P30530 1/20 0.37
MERTK Q12866 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29042039 1.00 IRAK4 (0.45) IRAK4GSK3BDYRK1AWNT1BMPR1B
SCHEMBL30508252 0.90 GSK3B (0.40) IRAK4GSK3BDYRK1AWNT1BMPR1B
SCHEMBL29041964 0.89 IRAK4 (0.48) IRAK4BMPR1BBMPR1ATGFBR1ACVRL1
SCHEMBL30508232 0.89 IRAK4 (0.48) IRAK4BMPR1BBMPR1ATGFBR1ACVRL1
SCHEMBL29042053 0.88 IRAK4 (0.42) IRAK4GSK3BDYRK1AWNT1BMPR1B
SCHEMBL30508229 0.88 IRAK4 (0.42) IRAK4GSK3BDYRK1AWNT1BMPR1B
SCHEMBL30508326 0.88 IRAK4 (0.42) IRAK4GSK3BDYRK1AWNT1BMPR1B
SCHEMBL29042061 0.83 BMPR1B (0.43) IRAK4GSK3BDYRK1AWNT1BMPR1B
SCHEMBL30508219 0.83 BMPR1B (0.43) IRAK4GSK3BDYRK1AWNT1BMPR1B
SCHEMBL30508339 0.77 MET (0.44) IRAK4BMPR1BBMPR1ATGFBR1ACVRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116478145-B ALK2 kinase inhibitors 杭州邦顺制药有限公司 2024-02-02 CN disclosed
CN-116478145-A ALK2 kinase inhibitors 杭州邦顺制药有限公司 2023-07-25 CN disclosed