SCHEMBL30509697

SCHEMBL30509697

C1=C(c2c[nH]c3ncccc23)CNCC12CC2

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.55
HTR2C P28335 1/20 0.55
HTR2B P41595 1/20 0.55
TGFBR1 P36897 3/20 0.44
PDPK1 O15530 2/20 0.44
IKBKE Q14164 2/20 0.44
CDC7 O00311 3/20 0.42
CDK2 P24941 3/20 0.42
CDK9 P50750 3/20 0.42
MAP4K4 O95819 2/20 0.42
PIM1 P11309 2/20 0.42
PRKACA P17612 2/20 0.42
GSK3B P49841 2/20 0.42
HIPK2 Q9H2X6 2/20 0.42
CLK4 Q9HAZ1 2/20 0.42
CDK5 Q00535 2/20 0.42
CCNT1 O60563 2/20 0.42
CCNA2 P20248 2/20 0.42
ROCK2 O75116 1/20 0.42
IRAK4 Q9NWZ3 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25428515 1.00 HTR2A (0.55) HTR2AHTR2CHTR2BTGFBR1PDPK1
Hydrochloric Acid SCHEMBL30509706 0.99 HTR2A (0.54) HTR2AHTR2CHTR2BTGFBR1PDPK1
Hydrochloric Acid SCHEMBL25428399 0.99 HTR2A (0.54) HTR2AHTR2CHTR2BTGFBR1PDPK1
SCHEMBL30509680 0.95 HTR2A (0.53) HTR2AHTR2CHTR2BTGFBR1PDPK1
SCHEMBL25426826 0.95 HTR2A (0.53) HTR2AHTR2CHTR2BTGFBR1PDPK1
SCHEMBL25865887 0.84 HTR2A (0.55) HTR2AHTR2CHTR2BTGFBR1PDPK1
SCHEMBL25865802 0.84 HTR2A (0.58) HTR2AHTR2CHTR2BTGFBR1PDPK1
Hydrochloric Acid SCHEMBL25428189 0.83 HTR2A (0.57) HTR2AHTR2CHTR2BTGFBR1PDPK1
Hydrochloric Acid SCHEMBL30509678 0.83 HTR2A (0.57) HTR2AHTR2CHTR2BTGFBR1PDPK1
SCHEMBL25865989 0.76 HTR2A (0.46) HTR2AHTR2CHTR2BTGFBR1PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4466266-B1 FUSED HETEROCYCLES AS 5-HT2A RECEPTOR AGONISTS TRANSNEURAL THERAPEUTICS INC (US) 2026-04-08 EP disclosed
US-12486268-B2 Fused heterocycles as 5-HT2A receptor agonists Transneural Therapeutics, Inc. (US) 2025-12-02 US disclosed
US-12459944-B2 Fused heterocycles as 5-HT2A receptor agonists Transneural Therapeutics, Inc. (US) 2025-11-04 US disclosed
US-20250243199-A1 FUSED HETEROCYCLES AS 5-HT2A RECEPTOR AGONISTS Transneural Therapeutics, Inc. (US) 2025-07-31 US disclosed
US-20240425503-A1 FUSED HETEROCYCLES AS 5-HT2A RECEPTOR AGONISTS Transneural Therapeutics, Inc. 2024-12-26 US disclosed
EP-4466266-A1 FUSED HETEROCYCLES AS 5-HT2A RECEPTOR AGONISTS Transneural Therapeutics, Inc. (US) 2024-11-27 EP disclosed
WO-2023141225-A1 FUSED HETEROCYCLES AS 5-HT2A RECEPTOR AGONISTS ONSERO THERAPEUTICS INC. (US) 2023-07-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12459944-B2 Fused heterocycles as 5-HT2A receptor agonists HTR2A, HTR2C, HTR5A HTR2A 1/4885HTR2C 2/4885HTR2B 6/4885
US-20250243199-A1 FUSED HETEROCYCLES AS 5-HT2A RECEPTOR AGONISTS HTR2A, HTR2C, HTR5A HTR2A 1/4885HTR2C 2/4885HTR2B 6/4885
US-20240425503-A1 FUSED HETEROCYCLES AS 5-HT2A RECEPTOR AGONISTS HTR2A, HTR2C, HTR1A HTR2A 1/4885HTR2C 2/4885HTR2B 6/4885
US-12486268-B2 Fused heterocycles as 5-HT2A receptor agonists HTR2A, HTR2C, HTR5A HTR2A 1/4885HTR2C 2/4885HTR2B 6/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.