SCHEMBL30515901

SCHEMBL30515901

COc1cc(Br)ccc1Oc1cccc(C)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.48
KMT2A Q03164 2/20 0.48
GAA P10253 1/20 0.48
FBP1 P09467 2/20 0.40
EGFR P00533 4/20 0.39
KDR P35968 2/20 0.39
TSHR P16473 3/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 2/20 0.39
LMNA P02545 2/20 0.39
TP53 P04637 1/20 0.39
ALOX15 P16050 1/20 0.39
CASP3 P42574 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
SENP6 Q9GZR1 1/20 0.39
ERBB2 P04626 2/20 0.39
ABCG2 Q9UNQ0 2/20 0.39
GAK O14976 1/20 0.39
MAPK13 O15264 1/20 0.39
ABL1 P00519 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24773597 1.00 KDM4E (0.48) KDM4EKMT2AGAAFBP1EGFR
SCHEMBL3197090 0.84 NPC1 (0.40) KDM4EFBP1EGFRKDRTSHR
SCHEMBL30366632 0.82 KDM4E (0.40) KDM4EKMT2AGAATSHRNPC1
SCHEMBL25715298 0.82 KDM4E (0.40) KDM4EKMT2AGAATSHRNPC1
SCHEMBL16695550 0.82 S1PR4 (0.37) KDM4EKMT2AGAATSHRNPC1
SCHEMBL4799459 0.82 LMNA (0.38) KDM4EKMT2AGAANPC1RAB9A
SCHEMBL4799471 0.82 KDM4E (0.44) KDM4EKMT2AGAAKDRTSHR
SCHEMBL28266977 0.80 ALDH1A1 (0.48) KDM4EKMT2ATSHRNPC1RAB9A
SCHEMBL25591263 0.75 PRKDC (0.59) KDM4EKMT2AGAAEGFRTSHR
SCHEMBL10548030 0.74 EGFR (0.44) KMT2AGAAEGFRKDRNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117886821-A Nitrogen-containing condensed ring derivative inhibitor, preparation method and application thereof 江苏豪森药业集团有限公司 2024-04-16 CN disclosed
CN-116514806-A Biological inhibitor containing acrylketone, preparation method and application thereof 上海翰森生物医药科技有限公司 2023-08-01 CN disclosed