SCHEMBL30516092

SCHEMBL30516092

CC(=O)c1cncc(-c2ncon2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK2 Q9HBH9 3/20 0.49
MKNK1 Q9BUB5 2/20 0.49
CYP11B2 P19099 5/20 0.43
CYP11B1 P15538 4/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
XDH P47989 2/20 0.40
PPARA Q07869 1/20 0.36
S1PR1 P21453 1/20 0.34
KAT6A Q92794 1/20 0.34
BRD4 O60885 2/20 0.33
BRD2 P25440 2/20 0.33
CREBBP Q92793 2/20 0.33
KMO O15229 1/20 0.33
MAP4K4 O95819 1/20 0.33
CSNK1G2 P78368 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
MAP4K5 Q9Y4K4 1/20 0.33
HCAR2 Q8TDS4 1/20 0.33
FYN P06241 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30516097 0.85 MKNK1 (0.47) MKNK2MKNK1XDHPPARAKMO
SCHEMBL30516103 0.83 ATM (0.51) CYP11B2CYP11B1S1PR1CYP2A6
SCHEMBL31364815 0.76 MKNK2 (0.54) MKNK2MKNK1CYP11B2CYP11B1CYP1A2
SCHEMBL29045118 0.74 CCNC (0.48) MKNK2MKNK1CYP11B2BRD4
SCHEMBL29045049 0.72 PPARA (0.40) PPARAKMO
SCHEMBL30516056 0.72 PPARA (0.40) PPARAKMO
SCHEMBL24921196 0.72 CYP1A1 (0.46) MKNK2MKNK1CYP11B2CYP11B1CYP1A2
SCHEMBL3500223 0.72 MKNK1 (0.55) MKNK2MKNK1CYP11B2CYP11B1CYP1A2
Hydrochloric Acid SCHEMBL30516112 0.71 PPARA (0.39) PPARAKMO
SCHEMBL4760887 0.70 PPARA (0.48) MKNK2MKNK1CYP11B2CYP11B1PPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116514790-A Tri-aromatic heterocyclic piperazine small molecular organic compound targeting STAT3 and application thereof 华东师范大学 2023-08-01 CN claimed
CN-116514790-A Tri-aromatic heterocyclic piperazine small molecular organic compound targeting STAT3 and application thereof 华东师范大学 2023-08-01 CN disclosed