SCHEMBL30516097

SCHEMBL30516097

O=C(O)c1cncc(-c2ncon2)c1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 1/20 0.47
MKNK2 Q9HBH9 1/20 0.47
HCAR2 Q8TDS4 5/20 0.44
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 3/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
POLB P06746 1/20 0.44
LMNA P02545 1/20 0.44
DDO Q99489 1/20 0.44
XDH P47989 1/20 0.38
KMO O15229 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
PPARA Q07869 1/20 0.37
EGLN1 Q9GZT9 1/20 0.35
CPT2 P23786 1/20 0.35
CPT1A P50416 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30516092 0.85 MKNK2 (0.49) MKNK1MKNK2HCAR2XDHKMO
SCHEMBL30516103 0.81 ATM (0.51) KDM4EALDH1A1
SCHEMBL3181717 0.78 MKNK1 (0.69) MKNK1MKNK2HCAR2KDM4EALDH1A1
SCHEMBL941077 0.77 KMO (0.53) KDM4EALDH1A1POLBKMO
SCHEMBL1319171 0.75 MKNK1 (0.53) MKNK1MKNK2HCAR2KDM4EALDH1A1
SCHEMBL15515155 0.75 TP53 (0.46) MKNK1MKNK2KDM4EALDH1A1
SCHEMBL29045118 0.75 CCNC (0.48) MKNK1MKNK2
SCHEMBL4760887 0.75 PPARA (0.48) MKNK1MKNK2KDM4EALDH1A1PPARA
SCHEMBL30516056 0.73 PPARA (0.40) KMOPPARA
SCHEMBL29045049 0.73 PPARA (0.40) KMOPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116514790-A Tri-aromatic heterocyclic piperazine small molecular organic compound targeting STAT3 and application thereof 华东师范大学 2023-08-01 CN disclosed