SCHEMBL30516699

SCHEMBL30516699

O=c1[nH]cnc2c(OCC(F)F)cc(-c3ccc(F)cn3)cc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.38
ACVR1 Q04771 2/20 0.36
FLT3 P36888 1/20 0.35
SYK P43405 1/20 0.35
AURKB Q96GD4 1/20 0.35
PDPK1 O15530 3/20 0.35
CHEK1 O14757 1/20 0.34
NTRK3 Q16288 2/20 0.34
MAPKAPK2 P49137 1/20 0.34
PNP P00491 1/20 0.34
NTRK1 P04629 1/20 0.34
IP6K1 Q92551 2/20 0.33
ROCK2 O75116 1/20 0.33
IP6K3 Q96PC2 1/20 0.33
BCL2 P10415 1/20 0.33
MCL1 Q07820 1/20 0.33
AURKA O14965 1/20 0.33
DAPK3 O43293 1/20 0.33
JAK2 O60674 1/20 0.33
PRKD3 O94806 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24478743 1.00 PARP1 (0.38) PARP1ACVR1FLT3SYKAURKB
SCHEMBL30516697 0.80 GRM5 (0.37) FLT3SYKAURKBNTRK3NTRK1
SCHEMBL24478613 0.80 GRM5 (0.37) FLT3SYKAURKBNTRK3NTRK1
SCHEMBL29631164 0.75 GRM5 (0.34) FLT3SYKAURKBNTRK3NTRK1
SCHEMBL22726094 0.71 PARP1 (0.50) PARP1ACVR1PDPK1CHEK1MAPKAPK2
SCHEMBL15845996 0.70 PDPK1 (0.57) PARP1PDPK1MAPKAPK2IP6K1IP6K3
Hydrochloric Acid SCHEMBL28036620 0.69 PDPK1 (0.56) PARP1PDPK1MAPKAPK2IP6K1IP6K3
SCHEMBL24478751 0.69 LDHA (0.42)
SCHEMBL30516696 0.69 LDHA (0.42)
SCHEMBL24478400 0.68 USP2 (0.35) AURKACLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116601149-A Aminoquinazoline derivatives as P2X3 inhibitors 奇斯药制品公司 2023-08-15 CN disclosed