Benzo[K]Tryptanthrin

Benzo[K]Tryptanthrin

SCHEMBL30537985

O=C1c2ccccc2-n2c1nc1cc3ccccc3cc1c2=O

nearest known ligand 0.71

Full drug profile on Sugi Atlas →

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 16/20 0.71
TDO2 P48775 15/20 0.71
IDO2 Q6ZQW0 13/20 0.71
NPC1 O15118 2/20 0.71
RAB9A P51151 2/20 0.71
KMT2A Q03164 2/20 0.71
LMNA P02545 1/20 0.71
NTRK1 P04629 1/20 0.71
ALOX5 P09917 1/20 0.71
MAPT P10636 1/20 0.71
PTGS2 P35354 1/20 0.71
HTT P42858 1/20 0.71
MAPK8 P45983 1/20 0.71
NTRK2 Q16620 1/20 0.71
HDAC6 Q9UBN7 1/20 0.71
APAF1 O14727 2/20 0.54
MEN1 O00255 1/20 0.54
MITF O75030 1/20 0.54
HSP90AA1 P07900 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzo[K]Tryptanthrin SCHEMBL9885118 1.00 IDO1 (0.71) IDO1TDO2IDO2NPC1RAB9A
SCHEMBL17830804 0.87 TDO2 (0.69) IDO1TDO2IDO2NPC1RAB9A
SCHEMBL18773427 0.86 IDO1 (0.68) IDO1TDO2IDO2NPC1RAB9A
SCHEMBL9100964 0.85 IDO1 (0.77) IDO1TDO2IDO2NPC1RAB9A
Tryptanthrin SCHEMBL2426211 0.83 TDO2 (1.00) IDO1TDO2IDO2NPC1RAB9A
Tryptanthrin SCHEMBL29359262 0.83 TDO2 (1.00) IDO1TDO2IDO2NPC1RAB9A
SCHEMBL30537967 0.83 TDO2 (0.74) IDO1TDO2IDO2NPC1RAB9A
SCHEMBL9101181 0.83 TDO2 (0.74) IDO1TDO2IDO2NPC1RAB9A
SCHEMBL9103139 0.83 TDO2 (0.74) IDO1TDO2IDO2NPC1RAB9A
SCHEMBL9103300 0.82 IDO1 (0.63) IDO1TDO2IDO2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4482584-A1 TRYPTANTHRIN DERIVATIVES WITH THIOSEMICARBAZONE SUBSTITUTION AND USE THEREOF Univerzita Karlova (CZ) 2025-01-01 EP disclosed
WO-2023160736-A1 TRYPTANTHRIN DERIVATIVES WITH THIOSEMICARBAZONE SUBSTITUTION AND USE THEREOF UNIVERZITA KARLOVA (CZ) 2023-08-31 WO disclosed