Tryptanthrin

Tryptanthrin

SCHEMBL29359262

O=C1c2ccccc2-n2c1nc1ccccc1c2=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 12/20 1.00
IDO2 Q6ZQW0 12/20 1.00
IDO1 P14902 11/20 1.00
KMT2A Q03164 3/20 1.00
LMNA P02545 3/20 1.00
NPC1 O15118 2/20 1.00
RAB9A P51151 2/20 1.00
HTT P42858 2/20 1.00
NTRK1 P04629 1/20 1.00
ALOX5 P09917 1/20 1.00
MAPT P10636 1/20 1.00
PTGS2 P35354 1/20 1.00
MAPK8 P45983 1/20 1.00
NTRK2 Q16620 1/20 1.00
HDAC6 Q9UBN7 1/20 1.00
APAF1 O14727 2/20 0.70
MEN1 O00255 2/20 0.70
MITF O75030 1/20 0.70
HSP90AA1 P07900 1/20 0.70
POLB P06746 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tryptanthrin SCHEMBL2426211 1.00 TDO2 (1.00) TDO2IDO2IDO1KMT2ALMNA
SCHEMBL9103006 0.84 TDO2 (1.00) TDO2IDO2IDO1KMT2ALMNA
SCHEMBL9101181 0.84 TDO2 (0.74) TDO2IDO2IDO1KMT2ALMNA
SCHEMBL30537967 0.84 TDO2 (0.74) TDO2IDO2IDO1KMT2ALMNA
SCHEMBL9103139 0.84 TDO2 (0.74) TDO2IDO2IDO1KMT2ALMNA
SCHEMBL12290069 0.84 IDO1 (0.80) TDO2IDO2IDO1KMT2ALMNA
SCHEMBL19456569 0.84 IDO1 (1.00) TDO2IDO2IDO1KMT2ALMNA
Benzo[K]Tryptanthrin SCHEMBL9885118 0.83 IDO1 (0.71) TDO2IDO2IDO1KMT2ALMNA
Benzo[K]Tryptanthrin SCHEMBL30537985 0.83 IDO1 (0.71) TDO2IDO2IDO1KMT2ALMNA
SCHEMBL9100596 0.83 APAF1 (1.00) TDO2IDO2IDO1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 467 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4615506-A1 USE OF GSK-3 ACTIVATIOR TO MODULATE PROTEASOME ACTIVITY TO PREVENT AGEING ASSOCIATED CONDITIONS AND DISEASES Sahin, Fikret (TR) 2025-09-17 EP claimed
US-20250171449-A1 TRYPTANTHRIN DERIVATIVES WITH THIOSEMICARBAZONE SUBSTITUTION AND USE THEREOF UNIVERZITA KARLOVA (CZ) 2025-05-29 US claimed
CN-119613411-A Method for synthesizing coupler aminoketone compound by photocatalysis and application 贵州大学 2025-03-14 CN claimed
CN-116655641-B Tryptamine ketimine compound and derivative thereof, and synthetic method and application thereof 成都大学 2025-03-11 CN claimed
CN-119462665-A 2-Fluoro-3-fatty amine tryptanthrin derivative, preparation method and application thereof 兴义民族师范学院 2025-02-18 CN claimed
CN-119462664-A 1,8 Disubstituted tryptanthrin derivative, preparation method and application thereof 兴义民族师范学院 2025-02-18 CN claimed
CN-119285637-A Tryptanthrin compound, synthesis method and application thereof 陕西中医药大学 2025-01-10 CN claimed
EP-4482584-A1 TRYPTANTHRIN DERIVATIVES WITH THIOSEMICARBAZONE SUBSTITUTION AND USE THEREOF Univerzita Karlova (CZ) 2025-01-01 EP claimed
WO-2024258363-A1 USE OF GSK-3 ACTIVATIOR TO MODULATE PROTEASOME ACTIVITY TO PREVENT AGEING ASSOCIATED CONDITIONS AND DISEASES SAHIN FIKRET (TR) 2024-12-19 WO claimed
CN-118766924-A Application of tryptanthrin in preparation of anti-colon cancer drugs 陕西中医药大学 2024-10-15 CN claimed
CN-114874220-A 8-aminobenzene sulfonamide substituted tryptanthrin derivative and preparation and application thereof 安徽瀚海博兴生物技术有限公司 2022-08-09 CN claimed
CN-114874219-A 2-aminobenzene sulfonamide substituted tryptanthrin derivative and preparation and application thereof 安徽瀚海博兴生物技术有限公司 2022-08-09 CN claimed
CN-113009035-B Method for identifying pharmacodynamic components of traditional Chinese medicine based on knocking out target components and application 福建卫生职业技术学院 2022-08-02 CN claimed
WO-2022094174-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF ESOPHAGEAL CONDITIONS CHILDREN'S HOSPITAL MEDICAL CENTER (US) 2022-05-05 WO claimed
CN-114206312-A Topical compositions and methods for treating inflammatory skin disorders 阿佐拉治疗股份有限公司 2022-03-18 CN claimed
WO-2022053964-A1 WATER-SOLUBLE TRYPTHANTRIN DERIVATIVES FOR REDOX FLOW BATTERIES UNIVERSIDADE DE COIMBRA (PT) 2022-03-17 WO claimed
CN-113016814-B Application of tryptanthrin derivative in treatment of plant virus and germ diseases 南开大学 2022-03-04 CN claimed
EP-3955889-A1 TOPICAL COMPOSITIONS AND METHODS FOR TREATING INFLAMMATORY SKIN DISEASES AZORA THERAPEUTICS, INC. (US) 2022-02-23 EP claimed
CN-113999231-A Alhaginine A derivative, preparation thereof and application thereof in preventing and treating plant virus and bacterial diseases 南开大学 2022-02-01 CN claimed
US-20220023259-A1 TOPICAL COMPOSITIONS AND METHODS FOR TREATING INFLAMMATORY SKIN DISEASES AZORA THERAPEUTICS, INC. 2022-01-27 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250171449-A1 TRYPTANTHRIN DERIVATIVES WITH THIOSEMICARBAZONE SUBSTITUTION AND USE THEREOF HTR3C, FTH1, GTF3C3 TDO2 18/4885IDO2 419/4885IDO1 406/4885
US-20220023259-A1 TOPICAL COMPOSITIONS AND METHODS FOR TREATING INFLAMMATORY SKIN DISEASES AHR, ARNT, TLR8 TDO2 38/4885IDO2 22/4885IDO1 15/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.