SCHEMBL30548975

SCHEMBL30548975

COC(=O)C1=Cc2cccnc2NC1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA12 O43570 6/20 0.42
CA9 Q16790 6/20 0.42
MAP2K1 Q02750 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.40
ALOX15 P16050 1/20 0.38
HTT P42858 1/20 0.38
KDM4E B2RXH2 4/20 0.38
TDP1 Q9NUW8 1/20 0.38
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37
MAPT P10636 1/20 0.37
CHRM3 P20309 1/20 0.36
HSD17B10 Q99714 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
CA2 P00918 1/20 0.36
CNR2 P34972 1/20 0.35
PKM P14618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28871698 0.85 POLB (0.36) TDP1ALDH1A1POLB
SCHEMBL5775122 0.81 KDM4E (0.38) L3MBTL1ALOX15KDM4ETDP1ALDH1A1
SCHEMBL29816028 0.81 KDM4E (0.38) L3MBTL1ALOX15KDM4ETDP1ALDH1A1
SCHEMBL30305190 0.80 PARP1 (0.36) KDM4EALDH1A1MAPTHSD17B10
SCHEMBL5779007 0.80 PARP1 (0.36) KDM4EALDH1A1MAPTHSD17B10
SCHEMBL27873839 0.79 L3MBTL1 (0.39) L3MBTL1KDM4ETDP1ALDH1A1MAPT
SCHEMBL26128039 0.77 CA12 (0.48) CA12CA9KDM4EALDH1A1POLB
SCHEMBL27726338 0.75 L3MBTL1 (0.44) CA12CA9MAP2K1L3MBTL1ALOX15
SCHEMBL29911876 0.71 TNKS2 (0.33) L3MBTL1ALDH1A1MAPT
SCHEMBL19142540 0.71 TNKS2 (0.33) L3MBTL1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023185811-A1 NOVEL HETEROCYCLIC COMPOUND 首药控股(北京)股份有限公司 2023-10-05 WO disclosed