SCHEMBL30554368

SCHEMBL30554368

c1ccc(C(c2ccccc2)(c2ccccc2)n2ncc3ccccc32)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.44
KMO O15229 1/20 0.40
CYP11B1 P15538 2/20 0.38
CYP11B2 P19099 2/20 0.38
CYP1A2 P05177 1/20 0.38
ADRA2A P08913 2/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
TFPI2 P48307 1/20 0.33
ASAH1 Q13510 1/20 0.33
KDM4E B2RXH2 2/20 0.33
SLC22A12 Q96S37 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
CASP1 P29466 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18113496 1.00 RECQL (0.44) RECQLKMOCYP11B1CYP11B2CYP1A2
SCHEMBL31540114 0.82 CYP11B1 (0.39) RECQLCYP11B1CYP11B2CYP1A2ADRA2A
SCHEMBL23901367 0.80 HDAC8 (0.41) KMOCYP11B1CYP11B2MEN1LMNA
SCHEMBL18113677 0.80 NR3C1 (0.32) CYP11B1CYP11B2
SCHEMBL20401326 0.80 ACSS2 (0.39) KDM4EMEN1ALDH1A1GAAMAPT
SCHEMBL9959744 0.77 ACSS2 (0.43) KDM4EALDH1A1HPGDKMT2ASMN1; SMN2
SCHEMBL29820308 0.76 CYP2A6 (0.39) KMOKDM4EMEN1ALDH1A1KMT2A
SCHEMBL12074315 0.76 HDAC8 (0.36) RECQL
SCHEMBL10050859 0.76 RECQL (0.43) RECQLKMOCYP11B1CYP11B2CYP1A2
SCHEMBL30449976 0.76 RECQL (0.43) RECQLKMOCYP11B1CYP11B2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024158745-A1 INHIBITORS OF LRRK2 VANDERBILT UNIVERSITY (US) 2024-08-02 WO disclosed
CN-112020357-B Salt of indazolyl-containing tricyclic derivative and crystal form thereof 上海翰森生物医药科技有限公司 2023-08-29 CN disclosed