SCHEMBL30558103

SCHEMBL30558103

COc1ccc(CN(Cc2ccc(OC)cc2)c2nc(Cl)ncc2[N+](=O)[O-])cc1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 10/20 0.49
MERTK Q12866 1/20 0.43
NPC1 O15118 3/20 0.42
DCTPP1 Q9H773 1/20 0.42
TXNRD1 Q16881 1/20 0.41
RAB9A P51151 2/20 0.40
KMT2A Q03164 2/20 0.40
PRKCQ Q04759 1/20 0.40
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28734428 0.90 PIN1 (0.43) PIN1MERTKNPC1DCTPP1RAB9A
SCHEMBL3787500 0.84 MERTK (0.59) MERTKNPC1DCTPP1TXNRD1ALDH1A1
SCHEMBL1560939 0.83 PIN1 (0.38) PIN1MERTKDCTPP1KMT2AALDH1A1
SCHEMBL30461993 0.80 LMNA (0.44) KMT2AALDH1A1LMNASMN1; SMN2
SCHEMBL11749778 0.76 PIN1 (0.45) PIN1ALDH1A1
SCHEMBL18757880 0.76 NPC1 (0.62) PIN1NPC1RAB9AKMT2APRKCQ
SCHEMBL4077793 0.75 PIN1 (0.47) PIN1ALDH1A1
SCHEMBL25381487 0.75 LMNA (0.47) NPC1DCTPP1RAB9AKMT2AALDH1A1
SCHEMBL1806718 0.75 PIN1 (0.77) PIN1MERTKALDH1A1LMNA
SCHEMBL29388790 0.74 PIK3CA (0.40) NPC1DCTPP1RAB9AKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116693458-A Cycloalkyl or heterocyclyl substituted heteroaryl compounds, compositions and uses thereof 深圳市塔吉瑞生物医药有限公司 2023-09-05 CN disclosed