SCHEMBL30558154

SCHEMBL30558154

[2H]C([2H])([2H])N1CCC(c2ccc(Br)cc2)CC1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
QDPR P09417 2/20 0.42
BRD4 O60885 1/20 0.41
SLC18A3 Q16572 2/20 0.40
LSS P48449 1/20 0.40
DRD2 P14416 2/20 0.38
MDM2 Q00987 1/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PRCP P42785 1/20 0.35
USP5 P45974 1/20 0.35
TSHR P16473 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL578267 0.86 QDPR (0.55) QDPRBRD4SLC18A3LSSDRD2
SCHEMBL999428 0.79 BRD4 (0.50) QDPRBRD4LSSMDM2CYP3A4
SCHEMBL21815500 0.79 BRD4 (0.50) QDPRBRD4LSSMDM2CYP3A4
SCHEMBL21205779 0.76 SLC18A3 (0.42) QDPRBRD4SLC18A3DRD2CYP3A4
SCHEMBL31222996 0.75 BRD4 (0.43) QDPRBRD4SLC18A3LSSDRD2
SCHEMBL265495 0.75 KDM1A (0.48) BRD4CYP3A4CYP2C9SMN1; SMN2
SCHEMBL14804315 0.75 KDM1A (0.48) BRD4CYP3A4CYP2C9SMN1; SMN2
SCHEMBL3469385 0.74 BRD4 (0.41) QDPRBRD4SLC18A3DRD2CYP3A4
SCHEMBL13677031 0.74 KCNH2 (0.49) BRD4SLC18A3DRD2MDM2CYP3A4
SCHEMBL6249416 0.74 DRD2 (0.53) SLC18A3DRD2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116693518-A Synthesis and application of EGFR inhibitor 江南大学 2023-09-05 CN disclosed