SCHEMBL30576754

SCHEMBL30576754

NC(=O)c1ccc(C=C2CCNCC2)cc1C(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.35
CRBN Q96SW2 1/20 0.34
APP P05067 1/20 0.33
ESRRA P11474 1/20 0.33
PARP1 P09874 1/20 0.32
NPFFR1 Q9GZQ6 2/20 0.32
NPFFR2 Q9Y5X5 2/20 0.32
MAPK10 P53779 1/20 0.32
GPR52 Q9Y2T5 1/20 0.31
PNMT P11086 1/20 0.31
CDC7 O00311 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC8 Q9BY41 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30576768 0.81 KMT2A (0.41) PARP1CDC7
SCHEMBL30576827 0.73 DHODH (0.48)
SCHEMBL26606446 0.73 DHODH (0.48)
SCHEMBL6071365 0.72 F2 (0.53)
SCHEMBL20567143 0.70 CHRM3 (0.51) PARP1
SCHEMBL30576800 0.70 FLT3 (0.42) PARP1
SCHEMBL30576808 0.69 PARP1 (0.36) PARP1PNMT
SCHEMBL30576779 0.68 ITGB3 (0.41) PARP1
SCHEMBL24177167 0.67 CES2 (0.47) CES2PARP1GPR52
SCHEMBL1002163 0.67 CES2 (0.72) CES2PARP1GPR52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116829542-A Benzothiazole and benzimidazole derivatives, pharmaceutically acceptable salts, preparation method thereof and pharmaceutical composition containing same as active ingredient 韩国化学研究院 2023-09-29 CN disclosed