SCHEMBL30586331

SCHEMBL30586331

c1cncc(OCCN2CCOCC2)c1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.78
CHRNA4 P43681 1/20 0.78
GAA P10253 1/20 0.60
NPC1 O15118 1/20 0.57
RAB9A P51151 1/20 0.57
EPHX2 P34913 1/20 0.57
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2D6 P10635 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
DRD2 P14416 3/20 0.56
DRD3 P35462 3/20 0.56
LTA4H P09960 2/20 0.56
CA12 O43570 1/20 0.55
CA1 P00915 1/20 0.55
CA2 P00918 1/20 0.55
CA7 P43166 1/20 0.55
CA9 Q16790 1/20 0.55
KDM4E B2RXH2 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13188216 0.93 CHRNB2 (0.67) CHRNB2CHRNA4GAAEPHX2CYP1A2
SCHEMBL7411609 0.88 CHRNB2 (1.00) CHRNB2CHRNA4DRD2DRD3LTA4H
SCHEMBL30601974 0.85 CHRNB2 (0.57) CHRNB2CHRNA4NPC1RAB9ACYP1A2
SCHEMBL6452945 0.82 NPC1 (0.79) NPC1RAB9ACYP1A2LTA4HCA12
Hydrochloric Acid SCHEMBL7013705 0.81 NPC1 (0.82) NPC1RAB9ALTA4HKDM4E
SCHEMBL14204567 0.81 NPC1 (0.77) NPC1RAB9ALTA4HCA12CA1
SCHEMBL14578276 0.80 ALDH1A1 (0.69) NPC1RAB9ALTA4HKDM4EALDH1A1
SCHEMBL20037920 0.79 NPC1 (0.60) GAANPC1RAB9ACYP1A2CYP3A4
SCHEMBL30422251 0.77 GAA (0.52) CHRNB2CHRNA4GAANPC1RAB9A
SCHEMBL3577214 0.77 TSHR (0.55) CHRNB2CHRNA4NPC1RAB9ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119317622-A Compounds useful as TYK2 inhibitors, preparation method and application thereof in medicine 上海致根医药科技有限公司 2025-01-14 CN disclosed
WO-2023165574-A1 COMPOUND USED AS TYK2 INHIBITOR, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL USE THEREOF 上海致根医药科技有限公司 2023-09-07 WO disclosed
CN-116693449-A Compounds useful as TYK2 inhibitors, preparation method and application thereof in medicine 上海致根医药科技有限公司 2023-09-05 CN disclosed