SCHEMBL30587607

SCHEMBL30587607

O=C(O)[C@H](CCCCO)N1C(=O)c2ccccc2C1=O

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.68
POLB P06746 4/20 0.68
KDM4E B2RXH2 1/20 0.68
TP53 P04637 1/20 0.68
GLA P06280 1/20 0.68
CYP3A4 P08684 1/20 0.68
CYP2D6 P10635 1/20 0.68
HPGD P15428 1/20 0.68
ALOX12 P18054 1/20 0.68
NFKB1 P19838 1/20 0.68
APEX1 P27695 1/20 0.68
MAPK1 P28482 1/20 0.68
HSD17B10 Q99714 1/20 0.68
GAA P10253 2/20 0.60
L3MBTL1 Q9Y468 2/20 0.50
HIF1A Q16665 1/20 0.50
DNMT1 P26358 6/20 0.48
KMT2A Q03164 3/20 0.48
CYP2C19 P33261 1/20 0.48
DNMT3B Q9UBC3 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5828004 1.00 ALDH1A1 (0.68) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL5828001 1.00 ALDH1A1 (0.68) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL6896852 0.89 ALDH1A1 (0.79) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL6896845 0.89 ALDH1A1 (0.79) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL3441076 0.86 ALDH1A1 (0.66) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL853260 0.86 ALDH1A1 (0.66) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL28775935 0.86 POLB (0.66) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL24130616 0.85 ALDH1A1 (0.64) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL31661829 0.85 POLB (0.64) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL21851961 0.85 ALDH1A1 (0.64) ALDH1A1POLBKDM4ETP53GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111269221-B Bicyclic lactams and methods of use thereof 豪夫迈·罗氏有限公司 2023-09-26 CN disclosed