SCHEMBL30592829

SCHEMBL30592829

COC(=O)c1ccc(OCc2c(-c3ccc(C)nc3)noc2C)nc1

nearest known ligand 0.79

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 12/20 0.79
GABRA5 P31644 8/20 0.78

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21403919 1.00 GABRA1 (0.79) GABRA1GABRA5
SCHEMBL29421368 0.93 GABRA5 (0.79) GABRA1GABRA5
SCHEMBL20241274 0.93 GABRA5 (0.79) GABRA1GABRA5
SCHEMBL30592886 0.93 GABRA5 (0.79) GABRA1GABRA5
SCHEMBL20241113 0.89 GABRA1 (0.82) GABRA1GABRA5
SCHEMBL30592788 0.89 GABRA1 (0.82) GABRA1GABRA5
SCHEMBL2924603 0.89 GABRA5 (0.84) GABRA1GABRA5
SCHEMBL20241313 0.89 GABRA1 (0.70) GABRA1GABRA5
SCHEMBL30592825 0.89 GABRA1 (0.70) GABRA1GABRA5
SCHEMBL20241395 0.88 GABRA1 (1.00) GABRA1GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117285525-A Novel isoxazolyl ether derivatives as GABAA alpha 5PAM 豪夫迈·罗氏有限公司 2023-12-26 CN disclosed
CN-109923113-B Isoxazolyl ether derivatives as GABA A alpha 5 PAM 豪夫迈·罗氏有限公司 2023-10-13 CN disclosed