SCHEMBL30593370

SCHEMBL30593370

Cc1cc(Br)cnc1N1CCN(C)CC1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 6/20 0.48
HRH3 Q9Y5N1 2/20 0.48
HTT P42858 1/20 0.47
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
NSD2 O96028 1/20 0.40
PKM P14618 1/20 0.40
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25406752 0.85 OPRK1 (0.50) HRH4HRH3
SCHEMBL30338745 0.85 OPRK1 (0.50) HRH4HRH3
SCHEMBL2366907 0.83 HRH4 (0.48) HRH4HTTMEN1CYP1A2CYP3A4
SCHEMBL19446958 0.82 HRH4 (0.48) HRH4MEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL1745337 0.82 KDM4E (0.36) HRH4HRH3ALDH1A1CYP3A4CYP2D6
SCHEMBL20605140 0.81 HRH4 (0.53) HRH4HRH3HTTSMN1; SMN2
SCHEMBL29969981 0.81 HRH4 (0.53) HRH4HRH3HTTSMN1; SMN2
SCHEMBL24970193 0.81 HRH4 (0.47) HRH4HRH3HTTALDH1A1CYP1A2
SCHEMBL1707795 0.81 ALDH1A1 (0.44) MEN1ALDH1A1CYP1A2CYP2C19KMT2A
SCHEMBL27829786 0.81 OPRK1 (0.37) HRH4HRH3ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116472047-B Arylamine derivative, preparation method and medical application thereof 中国医药研究开发中心有限公司 2025-06-17 CN disclosed
CN-116472047-A Arylamine derivative, preparation method and medical application thereof 中国医药研究开发中心有限公司 2023-07-21 CN disclosed