SCHEMBL30600809

SCHEMBL30600809

COc1cc(NC(=O)OC(C)(C)C)c2cnccc2c1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 1/20 0.43
CTSL P07711 2/20 0.41
CTSB P07858 1/20 0.41
NAMPT P43490 1/20 0.40
CYP17A1 P05093 3/20 0.40
CDC25B P30305 2/20 0.39
CLK1 P49759 1/20 0.39
CLK2 P49760 1/20 0.39
CLK3 P49761 1/20 0.39
CDK5 Q00535 1/20 0.39
DYRK1A Q13627 1/20 0.39
CDK5R1 Q15078 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
DYRK1B Q9Y463 1/20 0.39
MAPK14 Q16539 1/20 0.38
MAOA P21397 2/20 0.38
CYP3A4 P08684 1/20 0.37
KMT2A Q03164 1/20 0.37
SLC22A12 Q96S37 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30601010 0.85 MAP4K1 (0.44) MAP4K1NAMPTCYP17A1
SCHEMBL30600736 0.80 TRPV1 (0.51) NAMPTCDK5
SCHEMBL28365698 0.80 TRPV1 (0.51) NAMPTCDK5
SCHEMBL30600875 0.79 MAP4K1 (0.61) MAP4K1CYP17A1
SCHEMBL25859564 0.79 CLK1 (0.41) MAP4K1CTSLNAMPTCYP17A1CLK1
SCHEMBL38660013 0.78 MAP4K1 (0.51) MAP4K1NAMPTCYP17A1DYRK1ASLC22A12
SCHEMBL38659708 0.76 MAP4K1 (0.46) MAP4K1CYP17A1MAOAKMT2A
SCHEMBL26107591 0.75 CYP17A1 (0.52) NAMPTCYP17A1CLK1CLK2CLK3
SCHEMBL30596901 0.75 CYP17A1 (0.52) NAMPTCYP17A1CLK1CLK2CLK3
SCHEMBL23155544 0.75 NAMPT (0.46) NAMPTCYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110709392-B Isoquinoline as HPK1 inhibitor 豪夫迈·罗氏有限公司 2023-09-29 CN disclosed