SCHEMBL30603872

SCHEMBL30603872

CC(C)(C)OC(=O)N1CC=C(C#Cc2c(N)nc(N)nc2Cl)CC1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 8/20 0.55
TNK2 Q07912 2/20 0.40
GRM1 Q13255 5/20 0.39
ESR2 Q92731 1/20 0.38
PDK4 Q16654 1/20 0.37
NR1H2 P55055 1/20 0.37
BTK Q06187 1/20 0.37
JAK1 P23458 1/20 0.37
GPR119 Q8TDV5 1/20 0.36
CYP11B2 P19099 1/20 0.36
POLB P06746 1/20 0.36
ATR Q13535 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22476344 1.00 GRM5 (0.55) GRM5TNK2GRM1ESR2PDK4
SCHEMBL22476353 0.86 GRM5 (0.53) GRM5TNK2GRM1ESR2PDK4
SCHEMBL29110609 0.83 GRM5 (0.37) GRM5
SCHEMBL19971864 0.83 GRM5 (0.46) GRM5TNK2GRM1ESR2NR1H2
SCHEMBL941018 0.76 GRM5 (0.61) GRM5GRM1ESR2PDK4
SCHEMBL2893138 0.76 GRM5 (0.63) GRM5GRM1ESR2PDK4NR1H2
SCHEMBL3348910 0.75 GRM5 (0.66) GRM5GRM1ESR2PDK4JAK1
SCHEMBL19989696 0.74 GRM5 (0.69) GRM5GRM1ESR2PDK4GPR119
SCHEMBL14995149 0.73 GRM5 (0.70) GRM5GRM1ESR2PDK4GPR119
SCHEMBL20001581 0.73 GRM5 (0.60) GRM5GRM1ESR2PDK4NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116854709-A Reversible inhibitors of Bruton's tyrosine kinase and application thereof 药雅科技(上海)有限公司 2023-10-10 CN disclosed