SCHEMBL30604241

SCHEMBL30604241

COC(=O)c1cc(-c2ccc[nH]2)nc2ccccc12

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 1/20 0.66
DHODH Q02127 1/20 0.61
MEN1 O00255 6/20 0.59
KMT2A Q03164 6/20 0.59
KDM4E B2RXH2 9/20 0.58
ALDH1A1 P00352 7/20 0.58
HPGD P15428 4/20 0.58
TDP1 Q9NUW8 3/20 0.58
MAPK1 P28482 2/20 0.58
PKM P14618 2/20 0.58
LMNA P02545 2/20 0.58
PLIN1 O60240 1/20 0.58
GLA P06280 1/20 0.58
POLB P06746 1/20 0.58
PLIN5 Q00G26 1/20 0.58
MCL1 Q07820 1/20 0.58
ABHD5 Q8WTS1 1/20 0.58
MAPT P10636 4/20 0.57
TP53 P04637 2/20 0.57
L3MBTL1 Q9Y468 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13957934 0.85 KDM4E (0.63) TACR3DHODHMEN1KMT2AKDM4E
SCHEMBL30102549 0.85 KDM4E (0.63) TACR3DHODHMEN1KMT2AKDM4E
SCHEMBL14518623 0.85 MEN1 (0.72) DHODHMEN1KMT2AKDM4EALDH1A1
SCHEMBL30604083 0.83 TACR3 (0.57) TACR3DHODHMEN1KMT2AKDM4E
Bromide SCHEMBL4383984 0.82 MEN1 (0.69) DHODHMEN1KMT2AKDM4EALDH1A1
Hydrochloric Acid SCHEMBL4562712 0.82 MEN1 (0.69) TACR3DHODHMEN1KMT2AKDM4E
SCHEMBL2576382 0.81 KDM4E (0.76) TACR3DHODHMEN1KMT2AKDM4E
SCHEMBL6448659 0.80 TACR3 (1.00) TACR3MEN1KMT2AKDM4EALDH1A1
SCHEMBL14518625 0.80 MEN1 (0.66) DHODHMEN1KMT2AKDM4EALDH1A1
SCHEMBL30690048 0.78 DHODH (0.66) DHODHMEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116745291-A N- (2- (4-cyanothiazolidin-3-yl) -2-oxoethyl) -quinoline-4-carboxamide 阿斯利康(瑞典)有限公司 2023-09-12 CN disclosed