SCHEMBL30607708

SCHEMBL30607708

N#Cc1ccccc1-n1ncc2ccncc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCOA3 Q9Y6Q9 1/20 0.43
HTT P42858 1/20 0.43
KDM4E B2RXH2 1/20 0.42
CYP19A1 P11511 2/20 0.39
NR3C1 P04150 1/20 0.38
MAPT P10636 1/20 0.37
SLC2A1 P11166 1/20 0.37
SLC2A2 P11168 1/20 0.37
SLC2A3 P11169 1/20 0.37
PDE10A Q9Y233 1/20 0.36
CLK1 P49759 1/20 0.36
CLK2 P49760 1/20 0.36
CLK3 P49761 1/20 0.36
CDK5 Q00535 1/20 0.36
DYRK1A Q13627 1/20 0.36
CDK5R1 Q15078 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
DYRK1B Q9Y463 1/20 0.36
CSNK2A1 P68400 2/20 0.35
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30607673 0.73 PDE10A (0.39) MAPTPDE10A
SCHEMBL29833912 0.72 IRAK4 (0.53) KDM4EMAPTPDE10ACYP1A2
SCHEMBL30607638 0.70 NCOA3 (0.42) NCOA3HTTKDM4ECYP19A1CLK1
SCHEMBL31273773 0.68 MAOA (0.47) NCOA3HTTPDE10ACLK1CLK2
SCHEMBL29691131 0.67 KDM4E (0.64) KDM4ECYP19A1MAPTSLC2A1SLC2A2
SCHEMBL1671785 0.67 KDM4E (0.46) HTTKDM4ECYP19A1MAPTSLC2A1
SCHEMBL15839178 0.65 CYP17A1 (0.45) PDE10ACYP1A2
SCHEMBL27028753 0.65 MKNK2 (0.39) KDM4EPDE10ACYP1A2
SCHEMBL7015267 0.64 HTT (0.73) NCOA3HTTKDM4EMAPTPDE10A
SCHEMBL567999 0.64 CYP19A1 (0.57) CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023186065-A1 A CYCLIN-DEPENDENT KINASE INHIBITOR Taizhou Eoc Pharma Co., Ltd. (CN) 2023-10-05 WO disclosed