SCHEMBL30622467

SCHEMBL30622467

O=C(O)c1ccc2c(ccn2Cc2ccccn2)c1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 1/20 0.49
BRD4 O60885 1/20 0.47
KDM4E B2RXH2 1/20 0.46
SLC2A1 P11166 1/20 0.45
PPARG P37231 6/20 0.44
DRD4 P21917 1/20 0.44
CNR2 P34972 1/20 0.44
PLA2G4A P47712 1/20 0.43
EGFR P00533 1/20 0.43
ERBB2 P04626 1/20 0.43
ERBB4 Q15303 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31525423 0.85 EGFR (0.49) BRD4KDM4EPPARGEGFRERBB2
SCHEMBL30888879 0.81 PLAU (0.57) PPARG
SCHEMBL15971036 0.81 PLAU (0.57) PPARG
SCHEMBL6168536 0.80 KDM4E (0.52) KDM4CBRD4KDM4E
SCHEMBL31661504 0.79 SLC2A1 (0.54) BRD4SLC2A1EGFRERBB2ERBB4
SCHEMBL17067797 0.79 BRD4 (0.56) BRD4KDM4ESLC2A1EGFRERBB2
SCHEMBL3507524 0.79 SLC2A1 (0.54) BRD4SLC2A1EGFRERBB2ERBB4
SCHEMBL30622489 0.79 PLA2G4A (0.43) PPARGPLA2G4A
SCHEMBL6840362 0.77 PLG (0.53)
SCHEMBL11225244 0.77 CDK4 (0.53) BRD4SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250122152-A1 KAT6 Inhibitors BEIGENE SWITZERLAND GMBH (CH) 2025-04-17 US disclosed
WO-2025068943-A1 KAT6 INHIBITORS BEIGENE SWITZERLAND GMBH (CH) 2025-04-03 WO disclosed
US-20230330099-A1 SUBSTITUTED INDOLE MCL-1 INHIBITORS VANDERBILT UNIVERSITY 2023-10-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230330099-A1 SUBSTITUTED INDOLE MCL-1 INHIBITORS MCL1, BCL2L1, BCL9 KDM4C 2683/4885BRD4 71/4885KDM4E 1156/4885
US-20250122152-A1 KAT6 Inhibitors KAT6A, KAT6B, KAT7 KDM4C 1253/4885BRD4 303/4885KDM4E 948/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.