SCHEMBL30639503

SCHEMBL30639503

COc1cc(C(=O)O)c(OC[C@H](N)Cc2ccccc2)cn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN4A P35499 3/20 0.49
AKT1 P31749 9/20 0.43
TACR1 P25103 1/20 0.41
KLKB1 P03952 1/20 0.41
RPS6KB1 P23443 3/20 0.39
CHUK O15111 1/20 0.39
ROCK2 O75116 1/20 0.39
PIM1 P11309 1/20 0.39
PRKACA P17612 1/20 0.39
AKT2 P31751 1/20 0.39
CSNK1D P48730 1/20 0.39
GSK3A P49840 1/20 0.39
GSK3B P49841 1/20 0.39
PRKCD Q05655 1/20 0.39
ROCK1 Q13464 1/20 0.39
DYRK1A Q13627 1/20 0.39
CDC42BPA Q5VT25 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
PDPK1 O15530 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL27147895 0.95 SCN4A (0.44) SCN4AAKT1TACR1KLKB1RPS6KB1
SCHEMBL27032920 0.85 SCN4A (0.41) SCN4AAKT1TACR1KLKB1RPS6KB1
Trifluoroacetic Acid SCHEMBL29828724 0.84 SCN4A (0.41) SCN4AAKT1TACR1MEN1KMT2A
Trifluoroacetic Acid SCHEMBL29097359 0.84 SCN4A (0.41) SCN4AAKT1TACR1MEN1KMT2A
SCHEMBL27032995 0.78 SCN4A (0.48) SCN4AAKT1TACR1RPS6KB1PDPK1
SCHEMBL27133812 0.78 SCN4A (0.48) SCN4AAKT1TACR1RPS6KB1PDPK1
Hydrochloric Acid SCHEMBL27032816 0.77 SCN4A (0.49) SCN4AAKT1KLKB1RPS6KB1PDPK1
Hydrochloric Acid SCHEMBL27130904 0.77 SCN4A (0.49) SCN4AAKT1KLKB1RPS6KB1PDPK1
Hydrochloric Acid SCHEMBL27130810 0.75 AKT1 (0.49) SCN4AAKT1RPS6KB1CHUKROCK2
Hydrochloric Acid SCHEMBL27032824 0.75 AKT1 (0.49) SCN4AAKT1RPS6KB1CHUKROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116981672-A Macrocyclic compounds as CFTR modulators 爱杜西亚药品有限公司 2023-10-31 CN disclosed