SCHEMBL306442

SCHEMBL306442

CN(C)C1CCN(C(=O)c2cc3nccc(Oc4ccc(C(C(N)=O)C(=O)Nc5ccccc5)cc4F)c3s2)C1

nearest known ligand 0.74

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KDR P35968 20/20 0.74
MET P08581 19/20 0.74
MST1R Q04912 1/20 0.51
FLT1 P17948 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL307535 0.88 MET (0.71) KDRMET
SCHEMBL306443 0.85 MET (1.00) KDRMETMST1R
SCHEMBL304893 0.85 MET (1.00) KDRMETMST1R
SCHEMBL306678 0.83 MET (0.54) KDRMETMST1R
SCHEMBL307027 0.82 KDR (0.71) KDRMETMST1RFLT1
SCHEMBL307026 0.82 KDR (0.71) KDRMETMST1RFLT1
SCHEMBL16177167 0.80 KDR (0.77) KDRMETMST1RFLT1
SCHEMBL12251125 0.80 KDR (0.77) KDRMETMST1RFLT1
SCHEMBL307494 0.80 KDR (0.48) KDRMETFLT1
SCHEMBL308434 0.79 KDR (0.58) KDRMETFLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120083482-A1 INHIBITORS OF VEGF RECEPTOR AND HGF RECEPTOR SIGNALING METHYLGENE INC. 2012-04-05 US disclosed
US-8093264-B2 Fused heterocycles as inhibitors of VEGF receptor and HGF receptor signaling METHYLGENE INC. (CA) 2012-01-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120083482-A1 INHIBITORS OF VEGF RECEPTOR AND HGF RECEPTOR SIGNALING HGF, MET, KDR KDR 3/4885MET 2/4885MST1R 56/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.